Description
L-759,633 is a cannabinoid receptor 2 (CB2) selective agonist. It mimics CP 55,940 in a forskolin-induced cyclic AMP production assay by inhibiting the amount of cyclic AMP produced.
Product Unit Size | Cost | Quantity | Stock |
---|
L-759,633 is a cannabinoid receptor 2 (CB2) selective agonist. It mimics CP 55,940 in a forskolin-induced cyclic AMP production assay by inhibiting the amount of cyclic AMP produced.
Cas No. | 174627-50-0 |
---|---|
Purity | ≥98% |
Formula | C26H40O2 |
Formula Wt. | 384.60 |
Chemical Name | (6aR,10aR)-1-methoxy-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-6a,7,10,10a-tetrahydrobenzo[c]chromene |
IUPAC Name | (6aR,10aR)-1-methoxy-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-6a,7,10,10a-tetrahydrobenzo[c]chromene |
Solubility | 50mM in ethanol 25mM in DMSO |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Ross RA, Brockie HC, Stevenson LA, et al. Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656 and AM630. Br J Pharmacol. 1999 Feb;126(3):665-72. PMID: 10188977.
VEGFR inhibitor.
ERK1/2 inhibitor.
Nav1.7 and Nav1.8 N1+ channel blocker.
ITC found in cruciferous vegetables; AhR antago...
Fluoroquinolone; vacuolar H+ ATPase, topoisomer...
Dihydropyridine; L-type Ca2+ channel blocker.
Sulforaphane homolog, ITC found in cruciferous ...
Alliin analog found in cruciferous vegetables.<...
Macrolide antibiotic; peptidyl transferase inhi...
Aza-anthracenedione, DNA intercalator; topoisom...
Endogenous peptide involved in vascular contrac...
Endogenous opioid peptide; μOR agonist.
Isocitrate dehydrogenase inhibitor.
Selective 5-HT6 receptor antagonist
Oxidative phosphorylation inhibitor.
Alkaloid found in Corydalis; D1 antagonist, org...
Statin; HMG-CoA reductase inhibitor.
Fluoroquinolone, S-(-) isomer of ofloxacin; top...
EZH2 HMT inhibitor.
Cysteine-ITC conjugate, antioxidant.