Description
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
Product Unit Size | Cost | Quantity | Stock |
---|
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
Purity | ≥98% |
---|---|
Formula | C44H66N12O7S2 |
Formula Wt. | 939.2 |
Solubility | Soluble in water (2 mg/mL). |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Dooley CT, Chung NN, Schiller PW, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90(22):10811-5. PMID: 8248174.
Akt inhibitor.
HIV protease inhibitor, SERCA inhibitor.
β2-adrenergic agonist.
Roscovitine analog; CDK inhibitor.
Synthesis impurity
Pyrimidine, glucose analog, used to induce diab...
σ1/2and μ/κ/δ-OR agonist, α3β4/α4β2/α7...
Piperadine phenothiazine; FIASMA, D1-5, histami...
Flavanol originally found in Camilla (green tea...
Synthetic steroid hormone; glucocorticoid agoni...
Antimicrobial peptide found in frogs, induces p...
Alkaloid compound originally found in Corydalis...
Histamine H2 inverse agonist.
HIV and AIDS
Found in Piper longum; TxA2 antagonist, ubiquit...
Peptide fragment of VSV; LDLR agonist.
Aminocyclitol; protein synthesis inhibitor.
BH3 mimetic; Bcl-2 inhibitor.
Ras inhibitor.
Triterpene saponin found in Panax; Kv7.1 K+ cha...