Description
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
Product Unit Size | Cost | Quantity | Stock |
---|
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
Purity | ≥98% |
---|---|
Formula | C44H66N12O7S2 |
Formula Wt. | 939.2 |
Solubility | Soluble in water (2 mg/mL). |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Dooley CT, Chung NN, Schiller PW, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90(22):10811-5. PMID: 8248174.
Macrolide; peptidyl transferase inhibitor, prot...
Found in Evodia rutaecarpa; potential cAMP, 3β...
Thienylbutyl ITC analog.
Endogenous peptide, connects A and B chains of ...
Alkaloid found in species of Loranthus, Calia, ...
Endogenous catecholamine precursor, also found ...
Benzothiazepine; L-type Ca2+ channel blocker, p...
Nucleoside (guanosine) analog; DNA chain termin...
ITC.
D2 and 5-HT2A antagonist.
Sesquiterpene alcohol found in various essentia...
Zinc chelator
SIRT1 inhibitor.
Endogenous steroid hormone involved in reproduc...
T-type Ca2+ and voltage-gated Na+ channel block...
Fluoroquinolone; topoisomerase IV and bacterial...
Salicylic acid derivative; PPARγ agonist, pote...
Inhibitor of Monoacyglycerol lipase (MAGL).
Cysteine-ITC conjugate.
Dihydrofolate reductase inhibitor.