LKT Labs

Biochemicals for Life Science Research

KB-0742 dihydrochloride

KB-0742 dihydrochloride

Product ID K040009
Cas No. 2416874-75-2
Purity ≥99%
Product Unit SizeCostQuantityStock
1 mg $105.00 In stock
5 mg $193.00 In stock
10 mg $329.00 In stock
25 mg $579.00 In stock
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Description

KB-0742 dihydrochloride is a selective CDK9 inhibitor with potent anti-tumor activity in castration-resistant prostate cancer models.

Product Info

Cas No.

2416874-75-2
Purity

≥99%
Formula

C16H25N5 • 2HCl
Formula Wt.

360.32
IUPAC Name

(1S,3S)-3-N-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamine dihydrochloride
Synonym

KB0742 dihydrochloride, NSC-834161 dihydrochloride, NSC834161 dihydrochloride
Appearance

Yellow crystal powder

Shipping and Storage

Store Temp

-20°C
Ship Temp

Ambient

Downloads

Info Sheet

K040009 Info Sheet PDF

References

Richters A, Doyle S, Freeman D, et al. Modulating androgen receptor-driven transcription in prostate cancer with selective CDK9 inhibitors. Cell Chem Biol. 2021 Feb 18;28(2):134-147. PMID: 33086052

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