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Azaperone

Azaperone

Product ID A9801
Cas No. 1649-18-9
Purity ≥98%
Product Unit SizeCostQuantityStock
100 mg $127.90 In stock
500 mg $225.40 In stock
1 g $375.60 In stock
5 g $976.50 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Azaperone is a butyrophenone tranquilizer that exhibits sedative activity through the inhibition of α-adrenergic receptors. Azaperone also inhibits dopamine receptors and histamine receptors; it also may display antiemetic, antipsychotic, antihistaminergic, and anticholinergic activities.

Product Info

Cas No.

1649-18-9

Purity

≥98%

Formula

C19H22FN3O

Formula Wt.

327.40

Chemical Name

1-(4-Fluorophenyl)-4-[4-(2-pyridinyl)-1-piperazinyl]-1 -butanone

IUPAC Name

1-(4-fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one

Synonym

Stresnil, Suicalm

Melting Point

73-75°C

Solubility

Soluble in chloroform and ethyl acetate.

Appearance

A White or Almost White Crystalline Powder

Shipping and Storage

Store Temp

4°C

Ship Temp

Ambient

Downloads

MSDS

A9801 MSDS PDF

Info Sheet

A9801 Info Sheet PDF

References

Wolfe LL, Fisher MC, Davis TR, et al. Efficacy of a Low-Dosage Combination of Butorphanol, Azaperone, and Medetomidine (BAM) to Immobilize Rocky Mountain Elk. J Wildl Dis. 2014 Jul;50(3):676-80. PMID: 24807358.

McCormick AV, Wheeler JM, Guthrie CR, et al. Dopamine D2 receptor antagonism suppresses tau aggregation and neurotoxicity. Biol Psychiatry. 2013 Mar 1;73(5):464-71. PMID: 23140663.

Mentaberre G, López-Olvera JR, Casas-Díaz E, et al. Use of haloperidol and azaperone for stress control in roe deer (Capreolus capreolus) captured by means of drive-nets. Res Vet Sci. 2010 Jun;88(3):531-5. PMID: 20006891.

Leysen JE, Gommeren W. The dissociation rate of unlabelled dopamine antagonists and agonists from the dopamine-D2 receptor, application of an original filter method. J Recept Res. 1984;4(7):817-45. PMID: 6527363.

Custom Order

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