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Dermorphin

Dermorphin

Product ID D1769
Cas No. 77614-16-5
Purity ≥96%
Product Unit SizeCostQuantityStock
1 mg $189.00 Please Inquire
2 mg $325.50 In stock
5 mg $577.50 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Dermorphin is an opioid peptide originally found in the skin of amphibians; it exhibits analgesic and antinociceptive activities, acting as an agonist at μ-opioid receptors (μORs). In animal models of thermal, mechanical, and chemical pain, dermorphin increases pain thresholds.

Product Info

Cas No.

77614-16-5

Purity

≥96%

Formula

C40H50N8O10

Formula Wt.

802.88

Chemical Name

Tyrosyl-alanyl-phenylalanyl-glycyl-tyrosyl-prolyl-serinamide

IUPAC Name

(2S)-N-[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-[[2-[[(2S)-2- [[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl] amino]-3-phenylpropanoyl]amino]acetyl]amino]-3-(4-hydroxyphenyl) propanoyl]pyrrolidine-2-carboxamide

Solubility

Slightly soluble in water.

Appearance

White to off white powder

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

D1769 MSDS PDF

Info Sheet

D1769 Info Sheet PDF

References

Mizoguchi H, Bagetta G, Sakurada T, et al. Dermorphin tetrapeptide analogs as potent and long-lasting analgesics with pharmacological profiles distinct from morphine. Peptides. 2011 Feb;32(2):421-7. PMID: 21126548.

Guzevatykh LS, Voronina TA, Emel'ianova TG, et al. Comparative analysis of analgesic activities of dermorphin, [DPro6]-dermorphin, and their C-terminal tripeptides. Izv Akad Nauk Ser Biol. 2007 Sep-Oct;(5):577-82. PMID: 18038625.

Custom Order

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