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GSK-2982772

GSK-2982772

Product ID G733409
Cas No. 1622848-92-3
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $88.60 In stock
5 mg $170.40 In stock
25 mg $443.00 In stock
100 mg $1,083.40 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

GSK-2982772 is an inhibitor of receptor interacting protein 1 (RIP1), a regulator of necroptosis and inflammation. It has the potential to treat a variety of chronic inflammatory diseases such as psoriasis, rheumatoid arthritis, and ulcerative colitis.

Product Info

Cas No.

1622848-92-3

Purity

≥98%

Formula

C20H19N5O3

Formula Wt.

377.40

IUPAC Name

3-Benzyl-N-[(3S)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-1H-1,2,4-triazole-5-carboxamide

Synonym

GSK 2982772, GSK2982772

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

G733409 MSDS PDF

Info Sheet

G733409 Info Sheet PDF

References

Harris P., Berge S., et al. Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases. J Med Chem. 60(4):1247-61 (2017). PMID: 28151659.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
  • Total quantity of unit size desired (e.g. '10' in the case of 10 x 500 mg). If only one unit is desired, you may leave this blank.
  • This field is for validation purposes and should be left unchanged.

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