Description
Gusacitinib is a dual inhibitor of SYK/JAK kinases.
Product Unit Size | Cost | Quantity | Stock |
---|
Gusacitinib is a dual inhibitor of SYK/JAK kinases.
Cas No. | 1425381-60-7 |
---|---|
Purity | ≥98% |
Formula | C24H28N8O2 |
Formula Wt. | 460.54 |
IUPAC Name | 2-[1-[4-[4-(4-hydroxypiperidin-1-yl)anilino]-5-oxo-6H-pyrimido[4,5-d]pyridazin-2-yl]piperidin-4-yl]acetonitrile |
Synonym | ASN-002, ASN002 |
Appearance | Yellow powder |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
Info Sheet |
---|
Montilla A, Gomez-Garcia F, Gomez-Arias P, et al. Scoping review on the use of drugs targeting JAK/STAT pathway in atopic dermatitis, vitiligo, and alopecia areata. Dermatol The (Heidelb). 2019 Dec;9(4):655-683. PMID: 31606872
Inhibitor of Monoacyglycerol lipase (MAGL).
Hormonal attractant for male Bactrocera flies.<...
Peptide, involved in neutrophil activation; FPR...
Organosulfur, antioxidant.
Lignin found in Sesamin indicum;
Mycotoxin that has structural similarity to est...
Integrase inhibitor.
Endogenous hormone and neurotransmitter involve...
5-HT1B/1D agonist.
Pyrimidine nucleoside base, pairs with adenosin...
Polyether Ca2+ ionophore.
Selective inhibitor of the γ isoform of PI3K (...
Endogenous peptide hormone, involved in water h...
Dipeptide; aminopeptidase (N/CD13) inhibitor.
KRAS inhibitor
Flavonolignan mixture found in Silybum (milk th...
Peptide, derivative of AT I, cleavage product o...
Thrombin substrate used to measure thrombin act...
Recombinant Multi-epitope Chimeric HCV antigen....
Statin; HMG-CoA reductase inhibitor, potential ...