LKT Labs

Biochemicals for Life Science Research

MLN2480

MLN2480

Product ID M4452
Cas No. 1096708-71-2
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $123.00 In stock
5 mg $408.00 In stock
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Description

MLN2480 is an oral pan-Raf inhibitor designed to inhibit cell proliferation and survival. MLN2480 is currently in clinical trials and displays anticancer chemotherapeutic activity.

Product Info

Cas No.

1096708-71-2
Purity

≥98%
Formula

C17H12Cl2F3N7O2S
Formula Wt.

506.30
IUPAC Name

2-[(1R)-1-[(6-amino-5-chloropyrimidine-4-carbonyl)amino]ethyl]-N-[5- chloro-4-(trifluoromethyl)pyridin-2-yl]-1,3-thiazole-5-carboxamide
Solubility

DMSO 100 mg/mL (197.51 mM) Ethanol 100 mg/mL (197.51 mM) Water Insoluble

Shipping and Storage

Store Temp

-20°C
Ship Temp

Ambient

Downloads

MSDS

M4452 MSDS PDF
Info Sheet

M4452 Info Sheet PDF
Brochures

Ras-Raf-MEK-ERK Pathway Booklet

References

http://clinicaltrials.gov/show/NCT01425008

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