Name: BAY-1251152
SKU: B030962
Availability: InStock

Description

BAY-1251152 is an inhibitor of PTEFb/CDK9. PTEFb contributes to the regulation of gene transcription and can be over-expressed in cancer cells, leading to the transcription of key tumor-promoting genes and proliferation.

Product Info

Cas No.	1610358-56-9
Purity	≥98%
Formula	C₁₉H₁₈F₂N₄O₂S
Formula Wt.	404.44
IUPAC Name	5-Fluoro-4-(4-fluoro-2-methoxyphenyl)-N-{4-[(S-methylsulfonimidoyl)methyl]-2-pyridinyl}-2-pyridinamine
Synonym	BAY 1251152, BAY1251152

Shipping and Storage

Store Temp	-20°C
Ship Temp	Ambient

Downloads

MSDS	B030962 MSDS PDF
Info Sheet	B030962 Info Sheet PDF

References

Luecking U., Scholz A., et al. Identification of potent and highly selective PTEFb inhibitor BAY 1251152 for the treatment of cancer: from p.o. to i.v. application via scaffold hops. Cancer Res. 77(13 Suppl):Abstract nr 984 (2017).

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BAY-1251152

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