Description
CV-65 is a 1,8-Diaza-anthracene-tetrone compound that exhibits anticancer activity, inhibiting activation of JNK and ERK5 and suppressing proliferation in various tumor cell lines.
CV-65 is a 1,8-Diaza-anthracene-tetrone compound that exhibits anticancer activity, inhibiting activation of JNK and ERK5 and suppressing proliferation in various tumor cell lines.
| Purity | ≥70% |
|---|---|
| Formula | C14H10N2O4 |
| Formula Wt. | 270.24 |
| Chemical Name | 3,6-Dimethyl-1,8-diazaanthracene-2,7,9,10(1H,8H)-tetrone |
| IUPAC Name | 3,7-dimethyl-1,9-dihydropyrido[3,2-g]quinoline-2,5,8,10-tetrone |
| Appearance | Orange Solid |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet | |
| Brochures |
Pipaón C, Gutierrez P, Montero JC, et al. Mitogen-activated protein kinase routes as targets in the action of diaza-anthracene compounds with a potent growth-inhibitory effect on cancer cells. Mol Cancer Ther. 2002 Aug;1(10):811-9. PMID: 12492114.
CDK inhibitor.
Nucleoside (thymidine) analog; DNA chain termin...
Fluoroquinolone; topoisomerase IV and bacterial...
Methylxanthine; PDE inhibitor, A1/2 adenosine a...
mAChR agonist, selective for M2.
PI3K and PDK1 inhibitor.
Coumarin; VKORC1 inhibitor.
G-quadruplex ligand; DNA breakage inducer.
HIV protease inhibitor, SERCA inhibitor.
Endogenous peptide hormone inolved in gastric e...
Inhibitor of CDK.
Nav1.7 and Nav1.8 N1+ channel blocker.
Fast skeletal muscle troponin complex activator...
NSAID; COX inhibitor and HS-releasing agent.
Antimicrobial peptide found in amphibians.
Mast cell stabilizer; histamine H1/2/3 antagoni...
Kavalactone originally found in Piper methystic...
Endogenous biogenic amine, norepinephrine-like ...
Endogenous peptide, involved in immune signalin...
SIRT inhibitor.