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Deltarasin Hydrochloride Trihydrate

Deltarasin Hydrochloride Trihydrate

Product ID D1746
Cas No. 1440898-82-7
Purity ≥99%
Product Unit SizeCostQuantityStock
1 mg $112.60 In stock
5 mg $211.10 In stock
10 mg $329.30 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Deltarasin inhibits PDEδ at the farnesyl binding pocket, preventing its association with K-Ras. Deltarasin displays anticancer chemotherapeutic activity, inhibiting cell proliferation in cellular and animal models of pancreatic ductal adenocarcinoma.

Product Info

Cas No.

1440898-82-7

Purity

≥99%

Formula

C40H37N5O • xHCl • 3H2O

Formula Wt.

769.21

IUPAC Name

1-benzyl-2-[4-[(2S)-2-(2-phenylbenzimidazol-1-yl)-2-piperidin-4-ylethoxy]phenyl]benzimidazole;trihydrochloride; trihydrate

Solubility

DMSO 100 mg/mL (165.63 mM) Ethanol 100 mg/mL (165.63 mM) Water Insoluble

Appearance

White to off white powder

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

D1746 MSDS PDF

Info Sheet

D1746 Info Sheet PDF

References

Zimmermann G, Schultz-Fademrecht C, Küchler P, et al. Structure guided design and kinetic analysis of highly potent benzimidazole inhibitors targeting the PDEδ prenyl binding site. J Med Chem. 2014 Jun 26;57(12):5435-48. PMID: 24884780.

Zimmermann G, Papke B, Ismail S, et al. Small molecule inhibition of the KRAS-PDEδ interaction impairs oncogenic KRAS signalling. Nature. 2013 May 30;497(7451):638-42. PMID: 23698361.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
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