Description
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Product Unit Size | Cost | Quantity | Stock |
|---|
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Cas No. | 117830-79-2 |
|---|---|
| Purity | ≥97% |
| Formula | C21H86N3O6 |
| Formula Wt. | 496.57 |
| IUPAC Name | (2S)-2-[[(2S)-1-[2-[[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2- carbonyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-5- (diaminomethylideneamino)pentanoic acid |
| Synonym | APGPR; Procolipase activation peptide. |
| Solubility | Soluble in water (0.7 mg/mL). |
| Appearance | White to off-white powder |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Erlanson-Albertsson C. Fat-Rich Food Palatability and Appetite Regulation. In: Montmayeur JP, le Coutre J, editors. Fat Detection: Taste, Texture, and Post Ingestive Effects. Boca Raton (FL): CRC Press; 2010. Chapter 14. PMID: 21452478.
Takenaka Y, Shimano T, Mori T, et al. Enterostatin reduces serum cholesterol levels by way of a CCK(1) receptor-dependent mechanism. Peptides. 2008 Dec;29(12):2175-8. PMID: 18824202.
Lindqvist A, Berger K, Erlanson-Albertsson C. Enterostatin up-regulates the expression of the beta-subunit of F(1)F(o)-ATPase in the plasma membrane of INS-1 cells. Nutr Neurosci. 2008 Apr;11(2):55-60. PMID: 18510804.
Lignan found in Magnolia; GABA-A potentiator.
Endogenous peptide fragment, involved in vasoco...
ANP analog, cardiomodulatory peptide; NPR-A ago...
Endogenous sterol component of animal cell memb...
NO donor; AR antagonist.
Nucleoside (deoxyuridine) analog; DNA chain ter...
Synthetic peptide; FPRL1 agonist.
Steroid produced by Penicillum; PI3K, mTOR, DNA...
HDAC inhibitor.
Tretraeptide, binds cell surface integrins.
MET, VEGFR2, Ron, Axl, FLT3 inhibitor.
Endogenous hormone neurotransmitter, involved i...
Antimicrobial peptide found in Trichoderma, ind...
Peptide; GABA potentiator, NMDA negative allost...
Galactose analog, allolactose mimic, induces ac...
Fast skeletal muscle troponin complex activator...
Prenylated phenolic terpene found in various pl...
Thiazolidine macrolide found in the Red Sea spo...
S-enantiomer of citalopram; SERT inhibitor.
NSAID; COX-1/2 inhibitor.