Description
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Product Unit Size | Cost | Quantity | Stock |
|---|
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Cas No. | 117830-79-2 |
|---|---|
| Purity | ≥97% |
| Formula | C21H86N3O6 |
| Formula Wt. | 496.57 |
| IUPAC Name | (2S)-2-[[(2S)-1-[2-[[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2- carbonyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-5- (diaminomethylideneamino)pentanoic acid |
| Synonym | APGPR; Procolipase activation peptide. |
| Solubility | Soluble in water (0.7 mg/mL). |
| Appearance | White to off-white powder |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Erlanson-Albertsson C. Fat-Rich Food Palatability and Appetite Regulation. In: Montmayeur JP, le Coutre J, editors. Fat Detection: Taste, Texture, and Post Ingestive Effects. Boca Raton (FL): CRC Press; 2010. Chapter 14. PMID: 21452478.
Takenaka Y, Shimano T, Mori T, et al. Enterostatin reduces serum cholesterol levels by way of a CCK(1) receptor-dependent mechanism. Peptides. 2008 Dec;29(12):2175-8. PMID: 18824202.
Lindqvist A, Berger K, Erlanson-Albertsson C. Enterostatin up-regulates the expression of the beta-subunit of F(1)F(o)-ATPase in the plasma membrane of INS-1 cells. Nutr Neurosci. 2008 Apr;11(2):55-60. PMID: 18510804.
SARS-CoV-2 inhibitor
PKA inhibitor, potential ROCK, S6K1, MSK1, PKB ...
Nucleoside (guanosine) analog; DNA chain termin...
Anthraquinone found in aloe; CTFR Cl- channel a...
Fluoroquinolone; topoisomerase IV and bacterial...
Nitrobenzene; HPPD inhibitor.
Metabolite of spironolactone; Na+/K+ ATPase par...
Bioactive compound from olive tree.
Steroidogenesis inhibitor
Endogenous tripeptide, involved in HPA signalin...
Macrolide; protein translation inhibitor.
mTOR inhibitor.
Endogenous APP peptide cleavage product, primar...
Endogenous peptide, involved in paracrine and a...
KRAS inhibitor
Thiazide-like diuretic; Kv7.1 and minK K+ chann...
Rifampicin derivative; DNA-dependent RNA polyme...
Isoxazole derivative; HSP90 inhibitor.
ANP fragment, natriuretic peptide; Na+/K+ ATPas...
Glucocorticoid agonist.