Description
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Product Unit Size | Cost | Quantity | Stock |
|---|
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Cas No. | 117830-79-2 |
|---|---|
| Purity | ≥97% |
| Formula | C21H86N3O6 |
| Formula Wt. | 496.57 |
| IUPAC Name | (2S)-2-[[(2S)-1-[2-[[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2- carbonyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-5- (diaminomethylideneamino)pentanoic acid |
| Synonym | APGPR; Procolipase activation peptide. |
| Solubility | Soluble in water (0.7 mg/mL). |
| Appearance | White to off-white powder |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Erlanson-Albertsson C. Fat-Rich Food Palatability and Appetite Regulation. In: Montmayeur JP, le Coutre J, editors. Fat Detection: Taste, Texture, and Post Ingestive Effects. Boca Raton (FL): CRC Press; 2010. Chapter 14. PMID: 21452478.
Takenaka Y, Shimano T, Mori T, et al. Enterostatin reduces serum cholesterol levels by way of a CCK(1) receptor-dependent mechanism. Peptides. 2008 Dec;29(12):2175-8. PMID: 18824202.
Lindqvist A, Berger K, Erlanson-Albertsson C. Enterostatin up-regulates the expression of the beta-subunit of F(1)F(o)-ATPase in the plasma membrane of INS-1 cells. Nutr Neurosci. 2008 Apr;11(2):55-60. PMID: 18510804.
Selective inhibitor of c-Met.
Fibrate; PPARα agonist.
Folate analog; thymidylate synthase inhibitor.<...
Endogenous neuropeptide, also known as substanc...
Antioxidant, vitamin E derivative found in vege...
Tetracycline; protein translation inhibitor, MM...
Endogenous peptide hormone, involved in secreti...
Triterpene saponin found in species of Panax. <...
Trichothecene mycotoxin produced by Fusarium; p...
Dipeptide.
Broad-spectrum antibiotic
Vitamin B, required for formation of NAD and NA...
HIV protease inhibitor.
Endogenous cardiomodulatory peptide; NPR-A agon...
Coccidiostat, GAPDH inhibitor.
EZH2 HMT inhibitor.
Endogenous sulfonic acid involved in Ca2+ signa...
NSAID; COX-1/2 inhibitor.
Endogenous peptide hormone fragment, involved i...
Inhibitor of EGFR, HER2, VEGFR2, and FLT3.