Description
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Product Unit Size | Cost | Quantity | Stock |
|---|
Enterostatin is an endogenous anorexigenic peptide that regulates dietary fat intake and inhibits insulin secretion. Enterostatin binds the F1-ATPase β subunit and decreases serum cholesterol in a CCK-1 receptor-dependent manner.
| Cas No. | 117137-85-6 |
|---|---|
| Purity | ≥98% |
| Formula | C25H4N8O8 |
| Formula Wt. | 582.66 |
| IUPAC Name | 2-[[1-[2-[[1-(2-amino-3-methylbutanoyl)pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoic acid |
| Synonym | VPDPR |
| Solubility | Soluble in water. |
| Appearance | White to off-white powder |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Erlanson-Albertsson C. Fat-Rich Food Palatability and Appetite Regulation. In: Montmayeur JP, le Coutre J, editors. Fat Detection: Taste, Texture, and Post Ingestive Effects. Boca Raton (FL): CRC Press; 2010. Chapter 14. PMID: 21452478.
Takenaka Y, Shimano T, Mori T, et al. Enterostatin reduces serum cholesterol levels by way of a CCK(1) receptor-dependent mechanism. Peptides. 2008 Dec;29(12):2175-8. PMID: 18824202.
Lindqvist A, Berger K, Erlanson-Albertsson C. Enterostatin up-regulates the expression of the beta-subunit of F(1)F(o)-ATPase in the plasma membrane of INS-1 cells. Nutr Neurosci. 2008 Apr;11(2):55-60. PMID: 18510804.
Hec1/Nek2 mitotic pathway inhibitor
CDK2 inhibitor.
Neuraminidase inhibitor.
Fluoroquinolone; topoisomerase IV and bacterial...
BUB1 inhibitor.
Peptide, binds fibronectin.
FIASMA, SERT and DAT inhibitor, α1-adrenergic ...
Coenzyme, vitamin found in dairy, meat, eggs, f...
Minor kavalactone originally found in Piper met...
Nucleoside (adenosine) analog; viral DNA polyme...
Polymethoxy flavonoid found in citrus fruits.
Peptide, casein fragment.
Sulforaphane-cysteine conjugate.
NSAID; COX-1/2 inhibitor.
Synthetic antioxidant that induces phase II enz...
Peptide, alters uterine contractility; V1/2 and...
Bisphosphonate.
β1/2-adrenergic antagonist.
TRPV4 agonist
Nicotinic acid derivative; InhA inhibitor.