Description
Gusacitinib is a dual inhibitor of SYK/JAK kinases.
Product Unit Size | Cost | Quantity | Stock |
---|
Gusacitinib is a dual inhibitor of SYK/JAK kinases.
Cas No. | 1425381-60-7 |
---|---|
Purity | ≥98% |
Formula | C24H28N8O2 |
Formula Wt. | 460.54 |
IUPAC Name | 2-[1-[4-[4-(4-hydroxypiperidin-1-yl)anilino]-5-oxo-6H-pyrimido[4,5-d]pyridazin-2-yl]piperidin-4-yl]acetonitrile |
Synonym | ASN-002, ASN002 |
Appearance | Yellow powder |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
Info Sheet |
---|
Montilla A, Gomez-Garcia F, Gomez-Arias P, et al. Scoping review on the use of drugs targeting JAK/STAT pathway in atopic dermatitis, vitiligo, and alopecia areata. Dermatol The (Heidelb). 2019 Dec;9(4):655-683. PMID: 31606872
Pentacyclic triterpene found in the Banaba plan...
ITC found in cruciferous vegetables, analog of ...
AurKB/C inhibitor.
Endogenous pteridine metabolite of GTP.
SERCA inhibitor.
HDAC inhibitor. May reduce blood pressure in hy...
ATP-sensitive K+ channel activator, α-adrenerg...
PDE3 inhibitor.
GHB/GABA analog found in Valeriana officinalis;...
MEK1/2 inhibitor.
Steroid; AR antagonist.
Effective against gram-positive pathogens
Diaminoquinazoline derivative.
Inhibits NS5A
Flavonoid found in various plant sources; DAT a...
COVID-19 research
Endogenous peptide hormone involved in feeding ...
AChE inhibitor, D2 antagonist.
Peptide, derivative of AT II, involved in vasoc...
Fatty acid synthase inhibitor.