LKT Labs

Biochemicals for Life Science Research

MS436

MS436

Product ID M7200
Cas No. 1395084-25-9
Purity ≥99%
Product Unit SizeCostQuantityStock
1 mg $92.00 In stock
5 mg $179.00 In stock
25 mg $509.00 In stock
100 mg $1,048.00 In stock
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Description

MS346 is an inhibitor of bromodomain BRD4. This compound displays anti-inflammatory activity, decreasing the production of NO and pro-inflammatory cytokines in macrophages.

Product Info

Cas No.

1395084-25-9
Purity

≥99%
Formula

C18H17N5O3S
Formula Wt.

383.43
IUPAC Name

4-[(E)-(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-N-(2-pyridinyl)benzenesulfonamide
Solubility

100mM in DMSO

Shipping and Storage

Store Temp

-20°C
Ship Temp

Ambient

Downloads

MSDS

M7200 MSDS PDF
Info Sheet

M7200 Info Sheet PDF

References

Zhang G, Plotnikov AN, Rusinova E, et al. Structure-guided design of potent diazobenzene inhibitors for the BET bromodomains. J Med Chem. 2013 Nov 27;56(22):9251-64. PMID: 24144283.

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