Description
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
| Product Unit Size | Cost | Quantity | Stock |
|---|
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
| Purity | ≥98% |
|---|---|
| Formula | C44H66N12O7S2 |
| Formula Wt. | 939.2 |
| Solubility | Soluble in water (2 mg/mL). |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Dooley CT, Chung NN, Schiller PW, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90(22):10811-5. PMID: 8248174.
Alkylamine; histamine H1 antagonist, SERT and N...
Alkaloid found in plants in the Amaryllidaceae ...
FIASMA; α1- and β1/2-adrenergic antagonist.
Endogenous neuropeptide hormone, lowers extrace...
Heterocyclic light-emitting compound, natural l...
Adenosine analog
Respiratory toxin, mitochondrial permeability t...
ITC found in cruciferous vegetables; HDAC inhib...
Estradiol metabolite; microtubule depolymerizat...
Alters intracellular glutathione levels.
Synthetic antioxidant that induces phase II enz...
mAChR antagonist.
Bcl-2, Bcl-xl, sialyl transferase inhibitor.
Fast skeletal muscle troponin complex activator...
Fluoroquinolone; bacterial DNA gyrase inhibitor...
Aldose reductase inhibitor.
FK506 analog; calcineurin inhibitor.
Trichothecene mycotoxin produced by Fusarium.
Endogenous steroid hormone involved in immune r...
Allylbenzene found in spices and umbelliferous ...