Description
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
| Product Unit Size | Cost | Quantity | Stock |
|---|
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
| Purity | ≥98% |
|---|---|
| Formula | C44H66N12O7S2 |
| Formula Wt. | 939.2 |
| Solubility | Soluble in water (2 mg/mL). |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Dooley CT, Chung NN, Schiller PW, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90(22):10811-5. PMID: 8248174.
SMAC mimetic; PXR agonist, IAP inhibitor.
Macrolide antibiotic; peptidyl transferase inhi...
Mycotoxin produced by Fusarium; sphingosine acy...
Hydrophobic β-lactam; penicillin binding prote...
Semi-synthetic avermectin; GABA potentiator.
HDAC6 inhibitor.
FIASMA, SERT and NET inhibitor, mAChR antagonis...
Perfluorinated insecticide.
ITC found in cruciferous vegetables; AhR antago...
Ca2+ sensitizer; ATP-sensitive K+ channel activ...
A peroxisome proliferator-activated receptor ag...
Pyrimidine, glucose analog, used to induce diab...
Endogenous tachykinin peptide, involved in infl...
Impurity of rapamycin
MurA and isopentenyl mevalonate kinase inhibito...
Cathepsin K inhibitor.
c-MET inhibitor.
Selective cannabinoid receptor 2 (CB2) inverse ...
Voltage-gated Na+ channel blocker, mAChR antago...
Peptide found in amphibian skin; GRP (BB1) and ...