Description
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
| Product Unit Size | Cost | Quantity | Stock |
|---|
This acetalin peptide inhibits all opioid receptors with the greatest affinity for μ-opioid receptors (μORs) and the weakest affinity for δ-opioid receptors (δORs); it increases contractility in the guinea pig ileum assay.
| Purity | ≥98% |
|---|---|
| Formula | C44H66N12O7S2 |
| Formula Wt. | 939.2 |
| Solubility | Soluble in water (2 mg/mL). |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Dooley CT, Chung NN, Schiller PW, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90(22):10811-5. PMID: 8248174.
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