Description
RP-6306 is a protein kinase, membrane associated tyrosine/threonine 1 (PKMYT1) inhibitor.
| Product Unit Size | Cost | Quantity | Stock |
|---|
RP-6306 is a protein kinase, membrane associated tyrosine/threonine 1 (PKMYT1) inhibitor.
| Cas No. | 2719793-90-3 |
|---|---|
| Purity | ≥98% |
| Formula | C18H20N4O2 |
| Formula Wt. | 324.38 |
| Chemical Name | 2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethylpyrrolo[2,3-b]pyridine-3-carboxamide |
| IUPAC Name | 2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethylpyrrolo[2,3-b]pyridine-3-carboxamide |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| Info Sheet |
|---|
Chen J, Ren J, Zhang C, et al. Targeted delivery of the PKMYT1 inhibitor RP-6306 mediates PANoptosis in pancreatic cancer via mitotic catastrophe. Cell Death Dis. 2025 Jul 15;16(1):526. PMID: 40664640.
ITC, used as chiral agent.
Paclitaxel derivative
Curcumin derivative.
11β-HSD1 inhibitor.
LRRK2 inhibitor.
Monoterpene coumarin ether found in Citrus; PPA...
Alkaloid found in Corydalis and Stephania; D1/2...
Synthetic glucocorticoid
Inert clozapine analog, activates specialized G...
Fluoroquinolone; bacterial DNA gyrase inhibitor...
Synthetic ITC, erucin analog.
Voltage-gated Na+ channel blocker, mAChR antago...
EGFR inhibitor.
Endogenous peptide, produced by activation of P...
Carbapenem β-lactam; penicillin binding protei...
Recombinant Multi-epitope Chimeric HCV antigen....
Commercial food additive, antioxidant.
Benzazepine derivative; D1 partial agonist, pot...
Diterpene found in Anisomeles.
AMPK activator.