Description
RP-6306 is a protein kinase, membrane associated tyrosine/threonine 1 (PKMYT1) inhibitor.
| Product Unit Size | Cost | Quantity | Stock |
|---|
RP-6306 is a protein kinase, membrane associated tyrosine/threonine 1 (PKMYT1) inhibitor.
| Cas No. | 2719793-90-3 |
|---|---|
| Purity | ≥98% |
| Formula | C18H20N4O2 |
| Formula Wt. | 324.38 |
| Chemical Name | 2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethylpyrrolo[2,3-b]pyridine-3-carboxamide |
| IUPAC Name | 2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethylpyrrolo[2,3-b]pyridine-3-carboxamide |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| Info Sheet |
|---|
Chen J, Ren J, Zhang C, et al. Targeted delivery of the PKMYT1 inhibitor RP-6306 mediates PANoptosis in pancreatic cancer via mitotic catastrophe. Cell Death Dis. 2025 Jul 15;16(1):526. PMID: 40664640.
Inhibitor of EGFR, HER2, VEGFR2, and FLT3.
CDK4/6 inhibitor.
Endogenous opioid peptide; μOR agonist.
Thiazolidine; Pim kinase inhibitor.
Semi-synthetic analog of taxol; microtubule dep...
Endogenous peptide hormone, involved in stress ...
mAChR antaonist.
Calcium channel blocker.
Nucleoside (deoxyuridine) analog; DNA chain ter...
Endogenous neurotransmitter; GABA agonist.
Fluoroquinolone; topoisomerase IV, topoisomeras...
mTOR inhibitor.
Negative control for PKC activation.
Endogenous peptide hormone; GnRH agonist.
Triazole; 14-α demethylase inhibitor, potentia...
Fatty acid found in dairy products; HDAC inhibi...
Endogenous cardiomodulatory peptide; NPR-A agon...
Endogenous peptide hormone, GLP-1 fragment, inv...
5-HT1A agonist, 5-HT1B partial agonist, 5-HT3A/...
Cyclic peptide; calcineurin inhibitor.