Description
RP-6306 is a protein kinase, membrane associated tyrosine/threonine 1 (PKMYT1) inhibitor.
| Product Unit Size | Cost | Quantity | Stock |
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RP-6306 is a protein kinase, membrane associated tyrosine/threonine 1 (PKMYT1) inhibitor.
| Cas No. | 2719793-90-3 |
|---|---|
| Purity | ≥98% |
| Formula | C18H20N4O2 |
| Formula Wt. | 324.38 |
| Chemical Name | 2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethylpyrrolo[2,3-b]pyridine-3-carboxamide |
| IUPAC Name | 2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethylpyrrolo[2,3-b]pyridine-3-carboxamide |
| Store Temp | -20°C |
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| Ship Temp | Ambient |
| Info Sheet |
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Chen J, Ren J, Zhang C, et al. Targeted delivery of the PKMYT1 inhibitor RP-6306 mediates PANoptosis in pancreatic cancer via mitotic catastrophe. Cell Death Dis. 2025 Jul 15;16(1):526. PMID: 40664640.
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