Name: CEP-28122 Mesylate
SKU: C179604
Availability: InStock

Description

CEP-28122 is an ALK inhibitor. It inhibits tumor growth in ALK positive anaplastic large-cell lymphoma (ALCL), non-small cell lung cancer (NSCLC), and neuroglastoma cells.

Product Info

Cas No.	1354545-57-5
Purity	≥98%
Formula	C₂₈H₃₅ClN₆O₃ • CH₄O₃S
Formula Wt.	635.18
IUPAC Name	(1S,2S,3R,4R)-3-[(5-Chloro-2-{[(7S)-1-methoxy-7-(4-morpholinyl)-6,7,8,9-tetrahydro-5H-benzo[7]annulen-2-yl]amino}-4-pyrimidinyl)amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide methanesulfonate (1:1)
Synonym	CEP 28122 Mesylate, CEP28122 Mesylate
Solubility	10 mM in DMSO

Shipping and Storage

Store Temp	-20°C
Ship Temp	Ambient

Downloads

MSDS	C179604 MSDS PDF
Info Sheet	C179604 Info Sheet PDF

References

Cheng M., Quail M., et al. CEP-28122, a highly potent and selective orally active inhibitor of anaplastic lymphoma kinase with antitumor activity in experimental models of human cancers. Mol Cancer Ther. 11(3):670-79 (2012). PMID: 22203728.

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CEP-28122 Mesylate

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