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Eletriptan, Free Base

Eletriptan, Free Base

Product ID E4419
Cas No. 143322-58-1
Purity ≥90%
Product Unit SizeCostQuantityStock
1 mg $93.80 Please Inquire
5 mg $193.00 Please Inquire
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Eletriptan is a neuromodulator that acts an agonist at 5-HT1B/1D receptors and has selectivity for cranial arteries. Eletriptan is commonly used to treat acute migraines. Eletriptan inhibits activation of the trigeminovascular system, preventing nausea and emesis in vivo. Additionally, eletriptan may induce vasoconstriction of thoracic blood vessels, causing chest symptoms after administration.

Product Info

Cas No.

143322-58-1

Purity

≥90%

Formula

C22H26N2O2S

Formula Wt.

382.52

Chemical Name

3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-5-(2-phenylsulfonylethyl)-1H-indole

IUPAC Name

5-[2-(benzenesulfonyl)ethyl]-3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]- 1H-indole

Synonym

UK116044

Appearance

Yellowish Oil

Shipping and Storage

Store Temp

Ambient

Ship Temp

Ambient

Downloads

MSDS

E4419 MSDS PDF

Info Sheet

E4419 Info Sheet PDF

References

Almas M, Tepper SJ, Landy S, et al. Consistency of eletriptan in treating migraine: Results of a randomized, within-patient multiple-dose study. Cephalalgia. 2013 Dec 19. [Epub ahead of print]. PMID: 23946318.

Sandrini G, Perrotta A, Tassorelli C, et al. Eletriptan. Expert Opin Drug Metab Toxicol. 2009 Dec;5(12):1587-98. PMID: 19929447.

Wackenfors A, Jarvius M, Ingemansson R, et al. Triptans induce vasoconstriction of human arteries and veins from the thoracic wall. J Cardiovasc Pharmacol. 2005 May;45(5):476-84. PMID: 15821444.

Hoskin KL, Lambert GA, Donaldson C, et al. The 5-hydroxytryptamine1B/1D/1F receptor agonists eletriptan and naratriptan inhibit trigeminovascular input to the nucleus tractus solitarius in the cat. Brain Res. 2004 Feb 13;998(1):91-9. PMID: 14725972.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
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