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Mubritinib, Free Base

Product ID M8007
Cas No. 366017-09-6
Purity ≥99%
Product Unit SizeCostQuantityStock
5 mg $122.20 In stock
25 mg $489.00 In stock
100 mg $978.10 In stock
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  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Mubritinib is an EGFR2 (HER2) inhibitor that underwent clinical trials, showing some promise as an anticancer chemotherapeutic in the treatment of bladder, kidney, and prostate cancer, but was not pursued further.

Product Info

Cas No.

366017-09-6

Purity

≥99%

Formula

C25H23F3N4O2

Formula Wt.

468.47

Chemical Name

1-(4-{4-[(2-{(E)-2-[4-(trifluoromethyl)phenyl]ethenyl}-1,3-oxazol-4-yl)methoxy]phenyl}butyl)-1H-1,2,3-triazole

IUPAC Name

4-[[4-[4-(triazol-1-yl)butyl]phenoxy]methyl]-2-[(E)-2-[4- (trifluoromethyl)phenyl]ethenyl]-1,3-oxazole

Synonym

TAK-165

Appearance

White to off white powder

Shipping and Storage

Store Temp

Ambient

Ship Temp

Ambient

Downloads

MSDS

M8007 MSDS PDF

Info Sheet

M8007 Info Sheet PDF

References

Nagasawa J, Mizokami A, Koshida K, et al. Novel HER2 selective tyrosine kinase inhibitor, TAK-165, inhibits bladder, kidney and androgen-independent prostate cancer in vitro and in vivo. Int J Urol. 2006 May;13(5):587-92. PMID: 16771730.

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  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
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