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Picoplatin

Picoplatin

Product ID P3210
Cas No. 181630-15-9
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $173.70 In stock
5 mg $531.00 In stock
10 mg $837.20 In stock
25 mg $1,633.50 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Picoplatin is an analog of cisplatin with a 2-methylpyridine ligand that displays anticancer chemotherapeutic activity. Picoplatin is used to treat non-small cell lung cancer (NSCLC) and is in clinical trials as a potential treatment for prostate cancer. Picoplatin intercalates with GpG sequences in DNA and shows efficacy inhibiting tumor growth in vitro, in vivo, and in clinical settings.

Product Info

Cas No.

181630-15-9

Purity

≥98%

Formula

C6H10Cl2N2Pt

Formula Wt.

376.15

Chemical Name

azane; 2-methylpyridine; platinum(2+); dichloride

IUPAC Name

azane;2-methylpyridine;platinum(2+);dichloride

Appearance

White to pale yellow powder

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

P3210 MSDS PDF

Info Sheet

P3210 Info Sheet PDF

References

Matos CS, de Carvalho AL, Lopes RP, et al. New strategies against prostate cancer--Pt(II)-based chemotherapy. Curr Med Chem. 2012;19(27):4678-87. PMID: 22856665.

Eckardt JR, Bentsion DL, Lipatov ON, et al. Phase II study of picoplatin as second-line therapy for patients with small-cell lung cancer. J Clin Oncol. 2009 Apr 20;27(12):2046-51. PMID: 19289620.

Kanzawa F, Akiyama Y, Saijo N, et al. In vitro effects of combinations of cis-amminedichloro (2-methylpyridine) platinum (II) (ZD0473) with other novel anticancer drugs on the growth of SBC-3, a human small cell lung cancer cell line. Lung Cancer. 2003 Jun;40(3):325-32. PMID: 12781432.

Munk VP, Diakos CI, Ellis LT, et al. Investigations into the interactions between DNA and conformationally constrained pyridylamineplatinum(II) analogues of AMD473. Inorg Chem. 2003 Jun 2;42(11):3582-90. PMID: 12767196.

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