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Zafirlukast

Zafirlukast

Product ID Z0222
Cas No. 107753-78-6
Purity ≥98%
Product Unit SizeCostQuantityStock
10 mg $47.30 In stock
50 mg $189.30 In stock
100 mg $315.40 Please Inquire
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Zafirlukast is commonly recognized as a leukotriene receptor antagonist which is used in the treatment of asthma. It is found to be a potent inhibitor of VEGF-C/Nrp2. Research on topical usage suggests that zafirlukast may also be effective in preventing capsular contracture and reducing capsule formation of gel implants, a complication arising after breast implant surgery.

Product Info

Cas No.

107753-78-6

Purity

≥98%

Formula

C31H33N3O6S

Formula Wt.

575.68

Chemical Name

cyclopentyl N-[3-[[2-methoxy-4-[(2-methylphenyl)sulfonylcarbamoyl]phenyl]methyl]-1-methylindol-5-yl]carbamate

IUPAC Name

Cyclopentyl [3-(2-methoxy-4-{[(2-methylphenyl)sulfonyl]carbamoyl}benzyl)-1-methyl-1H-indol-5-yl]carbamate

Synonym

Accolate, Olmoran

Melting Point

138-140°C

Solubility

Soluble in DMSO (25 mg/ml).

Appearance

White to pink powder

Shipping and Storage

Store Temp

Ambient

Ship Temp

Ambient

Downloads

MSDS

Z0222 MSDS PDF

Info Sheet

Z0222 Info Sheet PDF

References

Oda S, Fijiwara R, Kutsuno Y, et al. Targeted screen for human UDP-glucuronosyltransferases inhibitors and the evaluation of potential drug-drug interactions with zafirlukast. Drug Metal Dispos. 2015 Jun; 43(6):812-818. PMID: 25834030.

Bandaru S, Marri VK, Kasera P, et al. Structure based virtual screening of ligands to identify cysteinyl leukotriene receptor 1 antagonist. Bioinformation. 2014 Oct 30; 10(10):652-657. PMID: 25489175.

Kang SH, Shin KC, Kim WS, et al. The preventive effect of topical zafirlukast instillation for peri-implant capsule formation in rabbits. Arch Plast Surg. 2015 Mar; 42(2):179-185. PMID: 25798389.

Custom Order

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