Description
Cyproterone is a steroidal anti-androgen that inhibits entry of androgens into the prostate. The acylated derivative of this compound is more potent and is used clinically more often.
| Product Unit Size | Cost | Quantity | Stock |
|---|
Cyproterone is a steroidal anti-androgen that inhibits entry of androgens into the prostate. The acylated derivative of this compound is more potent and is used clinically more often.
| Cas No. | 427-51-0 |
|---|---|
| Purity | ≥98% |
| Formula | C24H29ClO4 |
| Formula Wt. | 416.94 |
| Chemical Name | (1β,2β)-6-Chloro-1,2-dihydro-17-hydroxy-3'H- cyclopropa[1,2]pregna-1,4,6-triene-3,20-dione acetate |
| IUPAC Name | [(1S,2S,3S,5R,11R,12S,15R,16S)-15-acetyl-9-chloro-2,16-dimethyl-6-oxo-15-pentacyclo[9.7.0.02,8.03,5.012,16]octadeca-7,9-dienyl] acetate |
| Synonym | CPA, Androcur, Cyprostat |
| Melting Point | 200-201°C |
| Solubility | Soluble in dichloromethane and methyl alcohol. |
| Appearance | White or almost white crystalline powder |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Guadalix FJ, Botella Llusiá J. The action mechanism of cyproterone. Acta Ginecol (Madr). 1975 Jul 1;27(1):7-11. PMID: 1146472.
Giorgi EP, Shirley IM, Grant JK, et al. Androgen dynamics in vitro in the human prostate gland. Effect of cyproterone and cyproterone acetate. Biochem J. 1973 Mar;132(3):465-74. PMID: 4125095.
Chloramphenicol derivative; protein translation...
Potential VEGFR2, Met, RET, Axl, Ron, PDGFR, FG...
Polymixin, antimicrobial peptide, induces forma...
Polypeptide; peptidoglycan inhibitor.
Geldanamycin derivative; HSP90 inhibitor.
Abl, c-Kit, PDGFR inhibitor.
Steroidal jerveratrum alkaloid found in Veratru...
STING inhibitor
G-quadruplex ligand; DNA breakage inducer.
Bisphosphonate; FPPS inhibitor.
Ornithine decarboxylase inhibitor.
Derivative of methyl caffeate, hydroxycinnamic ...
c-MET inhibitor.
Selective Cannabinoid receptor 2(CB2) inverse a...
Semi-synthetic avermectin; GABA potentiator.
Phenothiazine derivative; D1/2 and 5-HT1A/2A an...
Endogenous neuropeptide hormone; somatostatin a...
Found in hawthorn.
Synthetic ITC.
Fatty acid synthase inhibitor.