Description
Amastatin inhibits enzymatic activity of aminopeptidases in vivo and in vitro; it also exhibits vasoconstrictive/pressor activity.
Amastatin Hydrochloride Hydrate
Product ID A4805
Cas No. 100938-10-1
Purity ≥98%
| Product Unit Size | Cost | Quantity | Stock |
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Product Info
| Cas No. | 100938-10-1 |
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| Purity | ≥98% |
| Formula | C21H38N4O8 • HCl • xH2O |
| Formula Wt. | 511.01 |
| IUPAC Name | 2-[[2-[[2-[(3-amino-2-hydroxy-5-methylhexanoyl)amino]-3-methylbutanoyl] amino]-3-methylbutanoyl]amino]butanedioic acid;hydrochloride |
| Synonym | [(2S,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl]-Val-Val-Asp-OH . HCl |
| Melting Point | 202-205°C |
| Solubility | Soluble in DMSO and acetic acid. |
| Appearance | White to off white powder |
Shipping and Storage
| Store Temp | 4°C |
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| Ship Temp | Ambient |
Downloads
| MSDS | |
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| Info Sheet |
References
Tobin VA, Arechaga G, Brunton PJ, et al. Oxytocinase in the female rat hypothalamus: a novel mechanism controlling oxytocin neurones during lactation. J Neuroendocrinol. 2014 Apr;26(4):205-16. PMID: 24612105.
Pillay D, Boulangé AF, Coustou V, et al. Recombinant expression and biochemical characterisation of two alanyl aminopeptidases of Trypanosoma congolense. Exp Parasitol. 2013 Dec;135(4):675-84. PMID: 24177338.
Batt CM, Klein EW, Harding JW, et al. Pressor responses to amastatin, bestatin and Plummer's inhibitors are suppressed by pretreatment with the angiotensin receptor antagonist sarthran. Brain Res Bull. 1988 Nov;21(5):731-5. PMID: 3219604.