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Amastatin Hydrochloride Hydrate

Amastatin Hydrochloride Hydrate

Product ID A4805
Cas No. 100938-10-1
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $75.10 In stock
5 mg $248.10 In stock
10 mg $435.80 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Amastatin inhibits enzymatic activity of aminopeptidases in vivo and in vitro; it also exhibits vasoconstrictive/pressor activity.

Product Info

Cas No.

100938-10-1

Purity

≥98%

Formula

C21H38N4O8 • HCl • xH2O

Formula Wt.

511.01

IUPAC Name

2-[[2-[[2-[(3-amino-2-hydroxy-5-methylhexanoyl)amino]-3-methylbutanoyl] amino]-3-methylbutanoyl]amino]butanedioic acid;hydrochloride

Synonym

[(2S,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl]-Val-Val-Asp-OH . HCl

Melting Point

202-205°C

Solubility

Soluble in DMSO and acetic acid.

Appearance

White to off white powder

Shipping and Storage

Store Temp

4°C

Ship Temp

Ambient

Downloads

MSDS

A4805 MSDS PDF

Info Sheet

A4805 Info Sheet PDF

References

Tobin VA, Arechaga G, Brunton PJ, et al. Oxytocinase in the female rat hypothalamus: a novel mechanism controlling oxytocin neurones during lactation. J Neuroendocrinol. 2014 Apr;26(4):205-16. PMID: 24612105.

Pillay D, Boulangé AF, Coustou V, et al. Recombinant expression and biochemical characterisation of two alanyl aminopeptidases of Trypanosoma congolense. Exp Parasitol. 2013 Dec;135(4):675-84. PMID: 24177338.

Batt CM, Klein EW, Harding JW, et al. Pressor responses to amastatin, bestatin and Plummer's inhibitors are suppressed by pretreatment with the angiotensin receptor antagonist sarthran. Brain Res Bull. 1988 Nov;21(5):731-5. PMID: 3219604.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
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