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Azilsartan

Azilsartan

Product ID A971334
Cas No. 147403-03-0
Purity ≥98%
Product Unit SizeCostQuantityStock
10 mg $90.20 In stock
50 mg $198.30 In stock
250 mg $390.60 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
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Description

Azilsartan is an angiotensin II receptor antagonist. It may provide a beneficial effect on the mechanisms involved in cardiometabolic disease and insulin sensitizing in cells. Diabetic mice treated with azilsartan had lowered expressions of pro-inflammatory cytokines in brain vessels and lowered diabetes-induced BBB permeability.

Product Info

Cas No.

147403-03-0

Purity

≥98%

Formula

C25H20N4O5

Formula Wt.

456.46

Chemical Name

2-ethoxy-3-[[4-[2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]phenyl]methyl]benzimidazole-4-carboxylic acid

IUPAC Name

2-ethoxy-3-[[4-[2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]phenyl]methyl]benzimidazole-4-carboxylic acid

Synonym

TAK-536; TAK 536

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

A971334 MSDS PDF

Info Sheet

A971334 Info Sheet PDF

References

Kurtz T, Kajiya T. Differential pharmacology and benefit/risk of azilsartan compared to other sartans. Vasc Health Risk Manag. 2012;8:133-143. PMID: 22399858.

Han J, Tang H, Yao L, et al. Azilsartan protects against hyperglycemia-induced hyperpermeability of the blood-brain barrier. Bioengineered. 2021 Dec;12(1):3621-3633. PMID: 34266350.

Li W, Wang C, Zhang D, et al. Azilsartan ameliorates ox-LDL-induced endothelial dysfunction via promoting the expression of KLF2. Aging (Albany NY). 2021 May 4; 13(9):12996-13005. PMID: 33946046.

Baker W, White W. Azilsartan medoxomil: a new angiotensin II receptor antagonist for treatment of hypertension. Ann Pharmacother. 2011 Dec;45(12):1506-1515. PMID: 22116996.

Custom Order

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