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BAY-1082439

BAY-1082439

Product ID B030960
Cas No. 1375469-38-7
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $81.70 In stock
5 mg $170.40 In stock
25 mg $497.60 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

BAY-1082439 is an inhibitor of PI3K. It is selective for the PI3Kα/β/δ isoforms. In vivo, BAY-1082439 has shown efficacy in inhibiting PTEN-null prostate cancer growth.

Product Info

Cas No.

1375469-38-7

Purity

≥98%

Formula

C25H30N6O5

Formula Wt.

494.55

IUPAC Name

N-{8-[(2R)-2-Hydroxy-3-(4-morpholinyl)propoxy]-7-methoxy-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl}-2-methylnicotinamide

Synonym

BAY 1082439, BAY1082439, BAY10-82439, BAY 10-82439, BAY-10-82439

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

B030960 MSDS PDF

Info Sheet

B030960 Info Sheet PDF

References

Zou Y., Qi Z., et al. Cotargeting the Cell-Intrinsic and Microenvironment Pathways of Prostate Cancer by PI3Kα/β/δ Inhibitor BAY1082439. Mol Cancer Ther. 17(10):2091-99 (2018). PMID: 30045927.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
  • Total quantity of unit size desired (e.g. '10' in the case of 10 x 500 mg). If only one unit is desired, you may leave this blank.
  • This field is for validation purposes and should be left unchanged.

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