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Cilostazol

Cilostazol

Product ID C3246
Cas No. 73963-72-1
Purity ≥98%
Product Unit SizeCostQuantityStock
10 mg $102.20 In stock
50 mg $277.60 In stock
100 mg $433.90 In stock
500 mg $1,323.00 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Cilostazol is a quinolone inhibitor of phosphodiesterase 3B (PDE 3B) that exhibits vasodilatory, antiplatelet, anti-inflammatory, anti-diabetic, antidepressant, anxiolytic, and pro-angiogenic activities. Cilostazol is clinically used to treat intermittent claudication associated with peripheral vascular disease. Cilostazol decreases production of TNF-α in macrophages and inhibits TNF-α-induced inflammation in adipose tissue, improving glucose tolerance and insulin resistance in vivo. Additionally, cilostazol decreases immobility time in the forced swim test and burying activity in the marble burying test. In other animal models, this compound upregulates production of G-CSF and VEGF, inducing angiogenesis.

Product Info

Cas No.

73963-72-1

Purity

≥98%

Formula

C20H27N5O2

Formula Wt.

369.46

Chemical Name

6-[4-(1-Cyclohexyl-1H-tetrazol-5-yl)-butoxy]-3,4- dihydro-2(1H)-quinolinone

IUPAC Name

6-[4-(1-cyclohexyltetrazol-5-yl)butoxy]-3,4-dihydro-1H-quinolin-2-one

Synonym

OPC-13013, Pletal

Melting Point

159.4-160.3°C

Solubility

Soluble in acetic acid, chloroform, and DMSO. Practically insoluble in water and ether.

Appearance

White to off white powder

Shipping and Storage

Store Temp

Ambient

Ship Temp

Ambient

Downloads

MSDS

C3246 MSDS PDF

Info Sheet

C3246 Info Sheet PDF

References

Biscetti F, Pecorini G, Straface G, et al. Cilostazol promotes angiogenesis after peripheral ischemia through a VEGF-dependent mechanism. Int J Cardiol. 2013 Aug 10;167(3):910-6. PMID: 22473072.

Wada T, Onogi Y, Kimura Y, et al. Cilostazol ameliorates systemic insulin resistance in diabetic db/db mice by suppressing chronic inflammation in adipose tissue via modulation of both adipocyte and macrophage functions. Eur J Pharmacol. 2013 May 5;707(1-3):120-9. PMID: 23528355.

Patel DS, Anand IS, Bhatt PA. Evaluation of antidepressant and anxiolytic activity of phosphodiesterase 3 inhibitor - cilostazol. Indian J Psychol Med. 2012 Apr;34(2):124-8. PMID: 23162186.

Custom Order

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