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CX-6258

CX-6258

Product ID C9200
Cas No. 1202916-90-2
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $98.00 In stock
5 mg $169.00 In stock
25 mg $540.00 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

CX-6258 is an inhibitor of Pim kinase that exhibits anticancer chemotherapeutic activity. This compound decreases tumor growth in animal models of cancer.

Product Info

Cas No.

1202916-90-2

Purity

≥98%

Formula

C26H24ClN3O3

Formula Wt.

461.95

IUPAC Name

(3E)-5-Chloro-3-[(5-{3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl}-2-furyl)methylene]-1,3-dihydro-2H-indol-2-one

Solubility

Water 89 mg/mL warmed (178.57 mM) DMSO 57 mg/mL warmed (114.36 mM) Ethanol 1 mg/mL warmed (2.0 mM)

Appearance

Light yellow solid

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

C9200 MSDS PDF

Info Sheet

C9200 Info Sheet PDF

References

Padmanabhan A, Gosc EB, Bieberich CJ. Stabilization of the prostate-specific tumor suppressor NKX3.1 by the oncogenic protein kinase Pim-1 in prostate cancer cells. J Cell Biochem. 2013 May;114(5):1050-7. PMID: 23129228.

Haddach M, Michaux J, Schwaebe MK, et al. Discovery of CX-6258. A Potent, Selective, and Orally Efficacious pan-Pim Kinases Inhibitor. ACS Med Chem Lett. 2011 Dec 27;3(2):135-9. PMID: 24900437.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
  • Total quantity of unit size desired (e.g. '10' in the case of 10 x 500 mg). If only one unit is desired, you may leave this blank.
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