Description
Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Product Unit Size | Cost | Quantity | Stock |
---|
Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Cas No. | 65189-71-1 |
---|---|
Purity | ≥95% |
Formula | C32H61N13O9 |
Formula Wt. | 771.92 |
IUPAC Name | 2-[[2-[[2-[2-[[2-[[2-[(2-amino-4-methylpentanoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]propanoylamino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]acetic acid |
Synonym | Phosphate Acceptor Peptide; NSC 332190. |
Solubility | Soluble in water (20 mg/mL), DMSO. |
Appearance | White to off white powder |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Montenegro M, Garcia-Viloca M, González-Lafont A, et al. Comparative study of the prereactive protein kinase A Michaelis complex with kemptide substrate. J Comput Aided Mol Des. 2007 Oct-Nov;21(10-11):603-15. PMID: 18008170.
Benyo DF, Zeleznik AJ. Cyclic adenosine monophosphate signaling in the primate corpus luteum: maintenance of protein kinase A activity throughout the luteal phase of the menstrual cycle. Endocrinology. 1997 Aug;138(8):3452-8. PMID: 9231800.
Whitehouse S, Feramisco JR, Casnellie JE, et al. Studies on the kinetic mechanism of the catalytic subunit of the cAMP-dependent protein kinase. J Biol Chem. 1983 Mar 25;258(6):3693-701. PMID: 6833226.
DOT1L HMT inhibitor.
Histamine H1 antagonist, FIASMA.
Triterpenoid found in Centella.
Nrf2-Keap1-ARE complex activator.
Cathepsin K inhibitor.
FIASMA, 5-HT1/2, M1-5 mAChR, α1-adrenergic, hi...
Bioactive compound from olive tree.
Isoxazole derivative; HSP90 inhibitor.
PI3K and mTOR inhibitor.
Endogenous opioid peptide derived from the β-c...
SIRT 1 activator, SIRT3 inhibitor.
Taxane found in Taxus; DNA polymerase inhibitor...
Chloramphenicol derivative; protein translation...
Src and Abl inhibitor.
Histamine H2 antagonist.
Synthetic peptide, stimulates gastric acid secr...
TrkB agonist.
Protein translation inhibitor.
5-HT2/3/6/7, D2/3/4, histamine H1, α1-adrenerg...