Description
Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Product Unit Size | Cost | Quantity | Stock |
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Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Cas No. | 65189-71-1 |
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Purity | ≥95% |
Formula | C32H61N13O9 |
Formula Wt. | 771.92 |
IUPAC Name | 2-[[2-[[2-[2-[[2-[[2-[(2-amino-4-methylpentanoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]propanoylamino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]acetic acid |
Synonym | Phosphate Acceptor Peptide; NSC 332190. |
Solubility | Soluble in water (20 mg/mL), DMSO. |
Appearance | White to off white powder |
Store Temp | -20°C |
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Ship Temp | Ambient |
MSDS | |
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Info Sheet |
Montenegro M, Garcia-Viloca M, González-Lafont A, et al. Comparative study of the prereactive protein kinase A Michaelis complex with kemptide substrate. J Comput Aided Mol Des. 2007 Oct-Nov;21(10-11):603-15. PMID: 18008170.
Benyo DF, Zeleznik AJ. Cyclic adenosine monophosphate signaling in the primate corpus luteum: maintenance of protein kinase A activity throughout the luteal phase of the menstrual cycle. Endocrinology. 1997 Aug;138(8):3452-8. PMID: 9231800.
Whitehouse S, Feramisco JR, Casnellie JE, et al. Studies on the kinetic mechanism of the catalytic subunit of the cAMP-dependent protein kinase. J Biol Chem. 1983 Mar 25;258(6):3693-701. PMID: 6833226.
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