Description
Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Product Unit Size | Cost | Quantity | Stock |
---|
Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Cas No. | 65189-71-1 |
---|---|
Purity | ≥95% |
Formula | C32H61N13O9 |
Formula Wt. | 771.92 |
IUPAC Name | 2-[[2-[[2-[2-[[2-[[2-[(2-amino-4-methylpentanoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]propanoylamino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]acetic acid |
Synonym | Phosphate Acceptor Peptide; NSC 332190. |
Solubility | Soluble in water (20 mg/mL), DMSO. |
Appearance | White to off white powder |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Montenegro M, Garcia-Viloca M, González-Lafont A, et al. Comparative study of the prereactive protein kinase A Michaelis complex with kemptide substrate. J Comput Aided Mol Des. 2007 Oct-Nov;21(10-11):603-15. PMID: 18008170.
Benyo DF, Zeleznik AJ. Cyclic adenosine monophosphate signaling in the primate corpus luteum: maintenance of protein kinase A activity throughout the luteal phase of the menstrual cycle. Endocrinology. 1997 Aug;138(8):3452-8. PMID: 9231800.
Whitehouse S, Feramisco JR, Casnellie JE, et al. Studies on the kinetic mechanism of the catalytic subunit of the cAMP-dependent protein kinase. J Biol Chem. 1983 Mar 25;258(6):3693-701. PMID: 6833226.
PDE3 inhibitor.
Aspirin analog; hemoglobin chain cross-linker.<...
Found in Aconitum bulleyanum; voltage-gated Na+...
Neurotoxin, mutagen.
Red-orange terpene pigment found in various pla...
B-Raf and c-Raf inhibitor.
Immunodominant peptide epitope occurring in mul...
Thiazolidinedione; PPARγ agonist.
Found in Magnolia officinalis.
Endogenous cardiomodulatory peptide; NPR-A agon...
Fibrate; PPARα agonist, enoyl-CoA reductase in...
Protein synthesis inhibitor, used to measure pr...
Selective inhibitor of cytochrome P450 1B1 (CYP...
Hydroxycinnamic acid found in coffee, argan oil...
Side chain attached to various taxanes.
Endogenous opioid peptide; μOR agonist.
Derivative of aristolochic acid found in Asarum...
Calpain I/II inhibitor.
Endogenous prostaglandin, vasodilator.
Viral RNA polymerase inhibitor.