Description
Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Product Unit Size | Cost | Quantity | Stock |
---|
Kemptide is a heptapeptide substrate of PKA used to measure PKA activity.
Cas No. | 65189-71-1 |
---|---|
Purity | ≥95% |
Formula | C32H61N13O9 |
Formula Wt. | 771.92 |
IUPAC Name | 2-[[2-[[2-[2-[[2-[[2-[(2-amino-4-methylpentanoyl)amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]propanoylamino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]acetic acid |
Synonym | Phosphate Acceptor Peptide; NSC 332190. |
Solubility | Soluble in water (20 mg/mL), DMSO. |
Appearance | White to off white powder |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Montenegro M, Garcia-Viloca M, González-Lafont A, et al. Comparative study of the prereactive protein kinase A Michaelis complex with kemptide substrate. J Comput Aided Mol Des. 2007 Oct-Nov;21(10-11):603-15. PMID: 18008170.
Benyo DF, Zeleznik AJ. Cyclic adenosine monophosphate signaling in the primate corpus luteum: maintenance of protein kinase A activity throughout the luteal phase of the menstrual cycle. Endocrinology. 1997 Aug;138(8):3452-8. PMID: 9231800.
Whitehouse S, Feramisco JR, Casnellie JE, et al. Studies on the kinetic mechanism of the catalytic subunit of the cAMP-dependent protein kinase. J Biol Chem. 1983 Mar 25;258(6):3693-701. PMID: 6833226.
Alkaloid found in Corydalis and Stephania; D1/2...
beta-Amyloid anti-oligomer and aggregation inhi...
Fluoroquinolone; topoisomerase IV and bacterial...
Antioxidant.
Marine toxin; actin polymerization inducer.
Selective 5-HT6 receptor antagonist
Selective inhibitor of the γ isoform of PI3K (...
Long chain acylcarnitine involved in fatty acid...
G-quadruplex ligand; DNA breakage inducer.
Macrolide lactone found in Bugula; TLR4 activat...
Sphingosine 1-phosphate antagonist.
Selective inhibitor of protein kinase C (PKC).<...
Ethisterone derivative, synthetic steroid, used...
mTOR inhibitor.
SERM.
Endogenous cardiomodulatory peptide; NPR-A agon...
D2 and D4 dopamine receptor inhibitor.
Found in plants in Astragalus, Allium, and Bras...
Nucleoside (thymidine) analog; DNA chain termin...
Hydroxycinnamic aicd, verbascoside metabolite, ...