Description
L-759,633 is a cannabinoid receptor 2 (CB2) selective agonist. It mimics CP 55,940 in a forskolin-induced cyclic AMP production assay by inhibiting the amount of cyclic AMP produced.
| Product Unit Size | Cost | Quantity | Stock |
|---|
L-759,633 is a cannabinoid receptor 2 (CB2) selective agonist. It mimics CP 55,940 in a forskolin-induced cyclic AMP production assay by inhibiting the amount of cyclic AMP produced.
| Cas No. | 174627-50-0 |
|---|---|
| Purity | ≥98% |
| Formula | C26H40O2 |
| Formula Wt. | 384.60 |
| Chemical Name | (6aR,10aR)-1-methoxy-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-6a,7,10,10a-tetrahydrobenzo[c]chromene |
| IUPAC Name | (6aR,10aR)-1-methoxy-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-6a,7,10,10a-tetrahydrobenzo[c]chromene |
| Solubility | 50mM in ethanol 25mM in DMSO |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Ross RA, Brockie HC, Stevenson LA, et al. Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656 and AM630. Br J Pharmacol. 1999 Feb;126(3):665-72. PMID: 10188977.
Cyclosporin metabolite; weak calmodulin inhibit...
Endogenous hormone involved in circadian rhythm...
Imidazole; 14-α demethylase inhibitor.
β-lactamase inhibitor.
Nucleoside (deoxycytidine) analog; DNMT inhibit...
Tripeptide, binds cell surface integrins.
Amphiphilic properties
Microtubule polymerization inhibitor.
FIASMA; α1- and β1/2-adrenergic antagonist.
p110α PI3K inhibitor.
NO donor; AR antagonist.
Peptide deformylase, MMP meprin A, aminopeptida...
Adenosine A2A agonist.
Natriuretic, vasodilatory peptide fragment; B1/...
Endogenous peptide fragment, involved in vasoco...
Hydrazine derivative, DNA alkylator; MAO inhibi...
Induces activation of Nrf2; inhibits apoptosis ...
Allosteric inhibitor
Phenyl hydrazide; neuronal oxidative stress inh...
Laminin-derived peptapeptide.