Description
LXS-196 is a selective inhibitor of protein kinase C (PKC). It is being investigated as a treatment for metastatic uveal melanoma, and may exhibit antitumor effects in other advanced tumors characterized by the overexpression of PKC.
| Product Unit Size | Cost | Quantity | Stock |
|---|
LXS-196 is a selective inhibitor of protein kinase C (PKC). It is being investigated as a treatment for metastatic uveal melanoma, and may exhibit antitumor effects in other advanced tumors characterized by the overexpression of PKC.
| Cas No. | 1874276-76-2 |
|---|---|
| Purity | ≥98% |
| Formula | C22H23F3N8O |
| Formula Wt. | 472.48 |
| Chemical Name | LXS-196 |
| IUPAC Name | 3-Amino-N-[3-(4-amino-4-methyl-1-piperidinyl)-2-pyridinyl]-6-[3-(trifluoromethyl)-2-pyridinyl]-2-pyrazinecarboxamide |
| Synonym | LXS 196, LXS196, NVP-LXS196, Darovasertib |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Wnt/beta-catenin/CBP inhibitor
Alternaria mycotoxin which may be found in food...
Taxane found in Taxus; potential microtubule de...
Metabolite of clofibrate; PPARα agonist.
ALK and IGF-1R inhibitor.
Glycopeptide, metal ion chelator, induces DNA s...
GPR84 agonist.
Phenyl hydrazide; neuronal oxidative stress inh...
Nucleoside (guanosine) analog; RT, guanylyl cyc...
ERK1/2 inhibitor.
PDE5 inhibitor.
Fluoroquinolone; topoisomerase IV and bacterial...
ROCK1/2 inhibitor, potential RSK and p70S6K inh...
Natriuretic, vasodilatory peptide, bradykinin a...
SIRT1/2 inhibitor, indirect p53 activator.
Polyphenol found in many plants and foods.
Recombinant BNP, cardiomodulatory peptide; NPR-...
H+/K+ ATPase and ROCK-2 inhibitor.
Endogenous peptide hormone fragment, involved i...
Anthracenedione, DNA intercalator; Pim-1 inhibi...