Description
LXS-196 is a selective inhibitor of protein kinase C (PKC). It is being investigated as a treatment for metastatic uveal melanoma, and may exhibit antitumor effects in other advanced tumors characterized by the overexpression of PKC.
| Product Unit Size | Cost | Quantity | Stock |
|---|
LXS-196 is a selective inhibitor of protein kinase C (PKC). It is being investigated as a treatment for metastatic uveal melanoma, and may exhibit antitumor effects in other advanced tumors characterized by the overexpression of PKC.
| Cas No. | 1874276-76-2 |
|---|---|
| Purity | ≥98% |
| Formula | C22H23F3N8O |
| Formula Wt. | 472.48 |
| Chemical Name | LXS-196 |
| IUPAC Name | 3-Amino-N-[3-(4-amino-4-methyl-1-piperidinyl)-2-pyridinyl]-6-[3-(trifluoromethyl)-2-pyridinyl]-2-pyrazinecarboxamide |
| Synonym | LXS 196, LXS196, NVP-LXS196, Darovasertib |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Mineralocorticoid antagonist.
Fibrate; PPARα agonist.
Kawain derivative, lactone found in Piper methy...
Nucleoside (thymidine) analog; DNA chain termin...
NO donor.
Aminoglycoside; protein translation inhibitor, ...
Thymidylate synthase inhibitor, potential SHMT,...
Saponin found in Polygala.
PDE3 inhibitor.
Triterpene saponin found in species of Panax.
May be useful against COVID-19
MDM2 inhibitor.
ITC precursor found in cruciferous vegetables.<...
ROCK1/2 inhibitor, potential RSK and p70S6K inh...
pan-PI3K inhibitor.
Folate source co-administered with methotrexate...
Water-soluble coenzyme, vitamin (B7) found in v...
mGluR5 positive modulator.
Terpene lactone found in Ginkgo.
Peptide, bee venom toxin; SK2/3/4 K+ channel bl...