Description
Telacebec is an imidazopyridine compound with high bactericidal activity. It may even be effective against extensively drug-resistant tuberculosis.
Product Unit Size | Cost | Quantity | Stock |
---|
Telacebec is an imidazopyridine compound with high bactericidal activity. It may even be effective against extensively drug-resistant tuberculosis.
Cas No. | 1334719-95-7 |
---|---|
Purity | ≥98% |
Formula | C29H28ClF3N4O2 |
Formula Wt. | 557.0 |
Chemical Name | 6-chloro-2-ethyl-N-[[4-[4-[4-(trifluoromethoxy)phenyl]piperidin-1-yl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide |
IUPAC Name | 6-chloro-2-ethyl-N-[[4-[4-[4-(trifluoromethoxy)phenyl]piperidin-1-yl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide |
Synonym | Q203, IAP6 |
Appearance | White powder |
Store Temp | 4°C |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Malik I, Cizmarik J, Kovac G, et al. Telacebec (Q203): Is there a novel effective and safe anti-tuberculosis drug on the horizon? Ceska Slov Farm. 2021 Winter;70(5):164-171. PMID: 35114793.
Lee B, Pethe K. Telacebec: an investigational antibacterial for the treatment of tuberculosis (TB). Expert Opin Investig Drugs. 2022 Feb;31(2):139-144. PMID: 35034512.
Komm O, Almeida D, Converse P, et al. Impact of dose, duration, and immune status on efficacy of ultrashort telacebec regimens in mouse models of Buruli ulcer. Antimicrob Agents Chemother. 2021 Oct 18;65(11):e0141821. PMID: 34460302.
5-Nitroimidazole derivative; genotoxic.
β-lactam; transpeptidase inhibitor.
Survivin inhibitor.
Antimuscarinic
Antiviral againt SARS-CoV-2
Furan derivative.
Tryptamine; 5-HT1B/1D agonist, TRPV1 antagonist...
Alkaloid compound originally found in Corydalis...
Indole, glucosinolate found in cruciferous vege...
Found in Salvia; MAG lipase inhibitor.
Flavonol glycoside originally found in Epimediu...
FIASMA, 5-HT3 and σ1 agonist, SERT inhibitor.<...
Kavalactone originally found in Piper methystic...
Orexin 2 receptor antagonist
Salicylic acid derivative; PPARγ agonist, pote...
Triazole; demethylation inhibitor.
Triterpene saponin found in Bupleurum.
Thiazolidinedione; PPARγ agonist.
Building block
Peptide fragment of HER2/neu/erbB2 receptor.