Description
Telacebec is an imidazopyridine compound with high bactericidal activity. It may even be effective against extensively drug-resistant tuberculosis.
Product Unit Size | Cost | Quantity | Stock |
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Telacebec is an imidazopyridine compound with high bactericidal activity. It may even be effective against extensively drug-resistant tuberculosis.
Cas No. | 1334719-95-7 |
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Purity | ≥98% |
Formula | C29H28ClF3N4O2 |
Formula Wt. | 557.0 |
Chemical Name | 6-chloro-2-ethyl-N-[[4-[4-[4-(trifluoromethoxy)phenyl]piperidin-1-yl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide |
IUPAC Name | 6-chloro-2-ethyl-N-[[4-[4-[4-(trifluoromethoxy)phenyl]piperidin-1-yl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide |
Synonym | Q203, IAP6 |
Appearance | White powder |
Store Temp | 4°C |
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Ship Temp | Ambient |
MSDS | |
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Info Sheet |
Malik I, Cizmarik J, Kovac G, et al. Telacebec (Q203): Is there a novel effective and safe anti-tuberculosis drug on the horizon? Ceska Slov Farm. 2021 Winter;70(5):164-171. PMID: 35114793.
Lee B, Pethe K. Telacebec: an investigational antibacterial for the treatment of tuberculosis (TB). Expert Opin Investig Drugs. 2022 Feb;31(2):139-144. PMID: 35034512.
Komm O, Almeida D, Converse P, et al. Impact of dose, duration, and immune status on efficacy of ultrashort telacebec regimens in mouse models of Buruli ulcer. Antimicrob Agents Chemother. 2021 Oct 18;65(11):e0141821. PMID: 34460302.
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