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Heptaplatin

Heptaplatin

Product ID H1862
Cas No. 146665-77-2
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $132.60 In stock
5 mg $301.70 In stock
10 mg $503.40 In stock
25 mg $956.00 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Heptaplatin is a platinum-complexed anticancer chemotherapeutic compound approved in some countries for the treatment of gastric cancers. Heptaplatin exhibits anti-proliferative activity in models of head and neck squamous cell cancers when combined with 5-fluorouracil (5-FU) as well as other, separate cancer cell lines.

Product Info

Cas No.

146665-77-2

Purity

≥98%

Formula

C11H20N2O6Pt

Formula Wt.

471.36

Chemical Name

[SP-4-2-[4R-(2a,4a,5b)]]-[2-(1-Methylethyl)-1,3-dioxolane-4,5-dimethanamine-N,N'][propanedioato(2-)-O,O']-platinum

IUPAC Name

[(4R,5R)-5-(aminomethyl)-2-propan-2-yl-1,3-dioxolan-4-yl]methanamine;platinum;propanedioic acid

Synonym

Eptaplatin

Appearance

White to off white powder

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

H1862 MSDS PDF

Info Sheet

H1862 Info Sheet PDF

References

Lee JW, Park JK, Lee SH, et al. Anti-tumor activity of heptaplatin in combination with 5-fluorouracil or paclitaxel against human head and neck cancer cells in vitro. Anticancer Drugs. 2006 Apr;17(4):377-84. PMID: 16549994.

Kim NK, Im SA, Kim DW, et al. Phase II clinical trial of SKI-2053R, a new platinum analog, in the treatment of patients with advanced gastric adenocarcinoma. Cancer. 1999 Oct 1;86(7):1109-15. PMID: 10506693.

Kim DK, Kim HT, Tai JH, et al. Pharmacokinetics and antitumor activity of a new platinum compound, cis-malonato[(4R,5R)-4,5-bis(aminomethyl)-2-isopropyl-1, 3- dioxolane]platinum(II), as determined by ex vivo pharmacodynamics. Cancer Chemother Pharmacol. 1995;37(1-2):1-6. PMID: 7497577.

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