Description
Urapidil is an α1-adrenergic receptor antagonist and 5-HT1A receptor agonist. Urapidil exhibits antihypertensive activity, inducing vasodilation and decreasing blood pressure without causing reflex tachycardia.
| Product Unit Size | Cost | Quantity | Stock |
|---|
Urapidil is an α1-adrenergic receptor antagonist and 5-HT1A receptor agonist. Urapidil exhibits antihypertensive activity, inducing vasodilation and decreasing blood pressure without causing reflex tachycardia.
| Cas No. | 34661-75-1 |
|---|---|
| Purity | ≥98% |
| Formula | C20H29N5O3 |
| Formula Wt. | 387.48 |
| Chemical Name | 6-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]- amino]-1,3-dimethyl-2,4(1H,3H)-pyrimidinedione |
| IUPAC Name | 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1, 3-dimethylpyrimidine-2,4-dione |
| Synonym | Ebrantil |
| Melting Point | 156-158°C |
| Solubility | Soluble in H2O. |
| Appearance | White Crystal Powder |
| Store Temp | Ambient |
|---|---|
| Ship Temp | Ambient |
| MSDS | |
|---|---|
| Info Sheet |
Santiveri X, Ledesma M. Urapidil in anesthesiology: pharmacology and indications. Rev Esp Anestesiol Reanim. 1998 May;45(5):189-97. PMID: 9646668.
van Zwieten PA, Chalmers JP. Different types of centrally acting antihypertensives and their targets in the central nervous system. Cardiovasc Drugs Ther. 1994 Dec;8(6):787-99. PMID: 7742257.
Found in Cladosporium; PKC inhibitor.
Methylated derivative of n-octyl-caffeate.
GRP analog, found in Bombina; bombesin and GRP ...
HDAC inhibitor. May reduce blood pressure in hy...
May induce apoptosis in lymphoma cell lines.
Triterpenoid
TLR4 inhibitor.
Imidazoquinoline nucleoside analog; TLR-7/8 ago...
Aminoglycoside; protein translation inhibitor, ...
Mycotoxin that has structural similarity to est...
GSK-3β inhibitor.
Impurity of omeprazole
p110α PI3K inhibitor.
Potential p53 activator or SIRT2 inhibitor.
JAK1/2 inhibitor.
Endogenous peptide fragment, involved in vasoco...
Somatostatin analog, peptide; somatostatin agon...
SERM.
Thiol prodrug, antioxidant.
AT1 inhibitor.