Description
Urapidil is an α1-adrenergic receptor antagonist and 5-HT1A receptor agonist. Urapidil exhibits antihypertensive activity, inducing vasodilation and decreasing blood pressure without causing reflex tachycardia.
Product Unit Size | Cost | Quantity | Stock |
---|
Urapidil is an α1-adrenergic receptor antagonist and 5-HT1A receptor agonist. Urapidil exhibits antihypertensive activity, inducing vasodilation and decreasing blood pressure without causing reflex tachycardia.
Cas No. | 34661-75-1 |
---|---|
Purity | ≥98% |
Formula | C20H29N5O3 |
Formula Wt. | 387.48 |
Chemical Name | 6-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]- amino]-1,3-dimethyl-2,4(1H,3H)-pyrimidinedione |
IUPAC Name | 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1, 3-dimethylpyrimidine-2,4-dione |
Synonym | Ebrantil |
Melting Point | 156-158°C |
Solubility | Soluble in H2O. |
Appearance | White Crystal Powder |
Store Temp | Ambient |
---|---|
Ship Temp | Ambient |
MSDS | |
---|---|
Info Sheet |
Santiveri X, Ledesma M. Urapidil in anesthesiology: pharmacology and indications. Rev Esp Anestesiol Reanim. 1998 May;45(5):189-97. PMID: 9646668.
van Zwieten PA, Chalmers JP. Different types of centrally acting antihypertensives and their targets in the central nervous system. Cardiovasc Drugs Ther. 1994 Dec;8(6):787-99. PMID: 7742257.
Laminin-derived peptapeptide.
Endogenous peptide hormone; CCK2 agonist, indir...
Wnt/β-catenin inhibitor
Chalcone kavalactone found in Piper methysticum...
HDAC inhibitor.
V600E B-Raf inhibitor.
Histamine H2 antagonist, GSK-3β inhibitor.
L-type Ca2+ channel blocker.
Peptide; GABA potentiator, NMDA negative allost...
Laminin-derived nonapeptide.
NSAID; COX-1/2 inhibitor.
Monoterpene; nAChR antagonist.
Mycotoxin produced by species of Aspergillus; D...
PRMT5 inhibitor
NO donor.
Endogenous peptide hormone, involved in feeding...
Found in propolis; 5-lipoxygenase inhibitor.
Derivative of methyl caffeate, hydroxycinnamic ...
c-Raf inhibitor, tyrosine kinase inhibitor.
AChE and BChE inhibitor.