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Vapreotide

Vapreotide

Product ID V0160
Cas No. 103222-11-3
Purity ≥95%
Product Unit SizeCostQuantityStock
0.5 mg $180.00 In stock
1 mg $306.70 In stock
2.5 mg $539.80 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Vapreotide is a synthetic peptide analog of somatostatin that activates somatostatin 2 receptors and inhibits neurokinin 1 receptors. Vapreotide exhibits anti-inflammatory, antiviral, orexigenic, antihypertensive, and anticancer chemotherapeutic activities. In macrophages, vapreotide inhibits substance P-induced production of IL-8 and MCP-1, preventing HIV-1 infection. In the clinical treatment of prostate cancer, vapreotide decreases PSA and PAP levels and bone pain scores. Additionally, this compound decreases portal pressure and blood flow, improving bleeding control and mortality rates in clinical subjects with variceal bleeding. Vapreotide also increases food intake in vivo.

Product Info

Cas No.

103222-11-3

Purity

≥95%

Formula

C57H70N12O9S2

Formula Wt.

1131.4

Chemical Name

L-Tryptophanamide, D-phenylalanyl-L-cysteinyl-L-tyrosyl-D- tryptophyl-L-lysyl-L-valyl-L-cysteinyl-, cyclic (2->7)-

IUPAC Name

(4R,7S,10S,13S,16S,19R)-10-(4-aminobutyl)-N-[(2R)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide

Synonym

Sanvar IR, BMY 41606, RC 160

Solubility

Soluble in water.

Appearance

White to off white powder

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

V0160 MSDS PDF

Info Sheet

V0160 Info Sheet PDF

References

Spitsin S, Tuluc F, Meshki J, et al. Analog of somatostatin vapreotide exhibits biological effects in vitro via interaction with neurokinin-1 receptor. Neuroimmunomodulation. 2013;20(5):247-55. PMID: 23921645.

Tachibana T, Cline MA, Khan MS, et al. Feeding responses to central administration of several somatostatin analogs in chicks. Comp Biochem Physiol A Mol Integr Physiol. 2011 Jan;158(1):47-51. PMID: 20826222.

Calès P. Vapreotide acetate for the treatment of esophageal variceal bleeding. Expert Rev Gastroenterol Hepatol. 2008 Apr;2(2):185-92. PMID: 19072353.

González-Barcena D, Schally AV, Vadillo-Buenfil M, et al. Response of patients with advanced prostatic cancer to administration of somatostatin analog RC-160 (vapreotide) at the time of relapse. Prostate. 2003 Aug 1;56(3):183-91. PMID: 12772187.

Custom Order

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