Description
AT-121 is a bifunctional agonist of the nociceptin/orphanin FQ peptide and mu opioid peptide receptors.
| Product Unit Size | Cost | Quantity | Stock |
|---|
AT-121 is a bifunctional agonist of the nociceptin/orphanin FQ peptide and mu opioid peptide receptors.
| Cas No. | 2099681-31-7 |
|---|---|
| Purity | ≥98% |
| Formula | C24H38N4O3S |
| Formula Wt. | 462.65 |
| Chemical Name | N-[2-[1,2-dihydro-1'-[cis-4-(1-methylethyl)cyclohexyl]-3-oxospiro[isoquinoline-4(3H),4'-piperidin]-2-yl]ethyl]-sulfamide 3-oxo-1'-(4-propan-2-ylcyclohexyl)-2-[2-(sulfamoylamino)ethyl]spiro[1H-isoquinoline-4,4'-piperidine] |
| IUPAC Name | 3-oxo-1'-(4-propan-2-ylcyclohexyl)-2-[2-(sulfamoylamino)ethyl]spiro[1H-isoquinoline-4,4'-piperidine] |
| Synonym | AT121 |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| Info Sheet |
|---|
Ding H, Kiguchi N, Yasuda D, et al. A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates. Sci Transl Med. 2018 Aug 29;10(456):eaar3483. PMID: 30158150.
Caffeic acid ester found in Melissa, Salvia, an...
PI3K inhibitor.
Neuropeptide hormone found in arthropods.
Benzophenanthridine alkaloid; topoisomerase I i...
Bisphosphonate, chelating agent.
Endogenous peptide hormone, involved in intesti...
First generation fluoroquinolone antibiotic.
Tyrphostin; VEGFR inhibitor.
FIASMA; α1- and β1/2-adrenergic antagonist.
Peptide, used as control to measure RGDS peptid...
Antimicrobial peptide found in Vespula lewisii,...
Antibiotic
Cephalosporin analogue
EGFR inhibitor.
Flavonoid found in species of Citrus; COX-2 inh...
Steroidal saponin found in Dioscorea.
BHA derivative.
Triterpene saponin originally found in Bolboste...
Peptide, used to tag proteins for affinity chro...
AKT inhibitor, potential ROCK, p70S6K, PKA, MKK...