Description
AT-121 is a bifunctional agonist of the nociceptin/orphanin FQ peptide and mu opioid peptide receptors.
| Product Unit Size | Cost | Quantity | Stock |
|---|
AT-121 is a bifunctional agonist of the nociceptin/orphanin FQ peptide and mu opioid peptide receptors.
| Cas No. | 2099681-31-7 |
|---|---|
| Purity | ≥98% |
| Formula | C24H38N4O3S |
| Formula Wt. | 462.65 |
| Chemical Name | N-[2-[1,2-dihydro-1'-[cis-4-(1-methylethyl)cyclohexyl]-3-oxospiro[isoquinoline-4(3H),4'-piperidin]-2-yl]ethyl]-sulfamide 3-oxo-1'-(4-propan-2-ylcyclohexyl)-2-[2-(sulfamoylamino)ethyl]spiro[1H-isoquinoline-4,4'-piperidine] |
| IUPAC Name | 3-oxo-1'-(4-propan-2-ylcyclohexyl)-2-[2-(sulfamoylamino)ethyl]spiro[1H-isoquinoline-4,4'-piperidine] |
| Synonym | AT121 |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| Info Sheet |
|---|
Ding H, Kiguchi N, Yasuda D, et al. A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates. Sci Transl Med. 2018 Aug 29;10(456):eaar3483. PMID: 30158150.
Butyrophenone; α-adrenergic, D2, histamine ant...
Cyclic peptide; calcineurin inhibitor.
Endogenous neuropeptide, somatostatin analog; s...
ITC, erucin analog.
Casein kinase 1 inhibitor.
Fetal hemoglobin stimulator; ribonucleotide red...
Viologen derivative
Hemantin inhibitor.
Micronuclei formation inducer, antimitotic, oxi...
Folic acid derivative
Tricyclic benzonaphthyridinone; mTORC1/2 inhibi...
Synthetic glycolipid found in Agelas mauritaniu...
Synthetic peptide hormone, PTH analog; PTH1R ag...
Tamoxifen derivative; potential proteasome inhi...
AChE inhibitor, F0F1-ATP synthase modulator.
Methylated derivative of n-octyl-caffeate.
Nucleoside (thymidine) analog; DNA chain termin...
ATP-sensitive K+ channel blocker, potential RyR...
Microtubule depolymerization inhibitor.
Chloramphenicol derivative; protein translation...