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AT-121

AT-121

Product ID A760010
Cas No. 2099681-31-7
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $450.00 Please Inquire
2 mg $800.00 Please Inquire
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Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

AT-121 is a bifunctional agonist of the nociceptin/orphanin FQ peptide and mu opioid peptide receptors.

Product Info

Cas No.

2099681-31-7

Purity

≥98%

Formula

C24H38N4O3S

Formula Wt.

462.65

Chemical Name

N-[2-[1,2-dihydro-1'-[cis-4-(1-methylethyl)cyclohexyl]-3-oxospiro[isoquinoline-4(3H),4'-piperidin]-2-yl]ethyl]-sulfamide 3-oxo-1'-(4-propan-2-ylcyclohexyl)-2-[2-(sulfamoylamino)ethyl]spiro[1H-isoquinoline-4,4'-piperidine]

IUPAC Name

3-oxo-1'-(4-propan-2-ylcyclohexyl)-2-[2-(sulfamoylamino)ethyl]spiro[1H-isoquinoline-4,4'-piperidine]

Synonym

AT121

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

Info Sheet

A760010 Info Sheet PDF

References

Ding H, Kiguchi N, Yasuda D, et al. A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates. Sci Transl Med. 2018 Aug 29;10(456):eaar3483. PMID: 30158150.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
  • Total quantity of unit size desired (e.g. '10' in the case of 10 x 500 mg). If only one unit is desired, you may leave this blank.
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