Description
Gusacitinib is a dual inhibitor of SYK/JAK kinases.
| Product Unit Size | Cost | Quantity | Stock |
|---|
Gusacitinib is a dual inhibitor of SYK/JAK kinases.
| Cas No. | 1425381-60-7 |
|---|---|
| Purity | ≥98% |
| Formula | C24H28N8O2 |
| Formula Wt. | 460.54 |
| IUPAC Name | 2-[1-[4-[4-(4-hydroxypiperidin-1-yl)anilino]-5-oxo-6H-pyrimido[4,5-d]pyridazin-2-yl]piperidin-4-yl]acetonitrile |
| Synonym | ASN-002, ASN002 |
| Appearance | Yellow powder |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| Info Sheet |
|---|
Montilla A, Gomez-Garcia F, Gomez-Arias P, et al. Scoping review on the use of drugs targeting JAK/STAT pathway in atopic dermatitis, vitiligo, and alopecia areata. Dermatol The (Heidelb). 2019 Dec;9(4):655-683. PMID: 31606872
Sartan
Imidazothiazole; alkaline phosphatase inhibitor...
Phosphodiesterase inhibitor that produces anti-...
Hec1/Nek2 mitotic pathway inhibitor
Cell membrane permeability modulator, topoisome...
Prolyl hydroxylase inhibitor.
Flavanol originally found in Camilla (green tea...
Recombinant HIV-1 antigen fragment.
AMPK activator, D1-4, 5-HT1A/2/3/6/7, M1-5 mACh...
GnRH analog; GnRH1 agonist.
Aminocyclitol; protein synthesis inhibitor.
Trichothecene mycotoxin produced by Fusarium; p...
Ester found in Spiraea, Betula, and Gaultheria;...
Thienopyridine; P2Y12 antagonist.
Vitamin E component
Calcium channel blocker.
Alkaloid found in Corydalis and Stephania; D1/2...
Tetracycline; protein translation inhibitor.
ACE inhibitor.
Highly selective inhibitor