Description
PF-04745637 is a selective antagonist for TRPA1 receptor.
Product Unit Size | Cost | Quantity | Stock |
---|
PF-04745637 is a selective antagonist for TRPA1 receptor.
Cas No. | 1917294-46-2 |
---|---|
Purity | ≥98% |
Formula | C27H32ClF3N2O2 |
Formula Wt. | 509.01 |
IUPAC Name | 1-(4-chlorophenyl)-N-[2-[4-hydroxy-4-(trifluoromethyl)piperidin-1-yl]-3-phenylpropyl]cyclopentane-1-carboxamide |
Appearance | White solid |
Store Temp | -20°C |
---|---|
Ship Temp | Ambient |
Info Sheet |
---|
p110γ PI3K inhibitor.
CDK1/2 inhibitor.
FIASMA; α1- and β1/2-adrenergic antagonist.
5-HT3 antagonist.
Cembranoid found in Sarcophyton.
Sialic-acid sensing lectin.
DOT1L HMT inhibitor.
VEGF-C/Nrp2 inhibitor. Leukotriene receptor ant...
Benzazepine derivative; D1 partial agonist, pot...
Triazole; 14α demethylase inhibitor.
FIASMA, mAChR, 5-HT2/3/6/7, α1/2-adrenergic an...
Endogenous peptide hormone, involved in stress ...
Prenylated phenolic terpene found in various pl...
Synthesis intermediate
Water-soluble parthenolide analog; NF-κB inhib...
Aza-anthracenedione, DNA intercalator; topoisom...
FAK inhibitor.
TRPA1 agonist, xanthine oxidase inhibitor.
Neuroactive mycotoxin produced by Penicillum an...
Melatonin analog; MT1/2 agonist, 5-HT2C antagon...