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Azilsartan Medoxomil

Azilsartan Medoxomil

Product ID A971336
Cas No. 863031-21-4
Purity ≥98%
Product Unit SizeCostQuantityStock
5 mg $93.80 In stock
25 mg $294.50 In stock
100 mg $691.00 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Azilsartan medoxomil is an angiotensin II receptor antagonist. It may provide a beneficial effect on the mechanisms involved in cardiometabolic disease and insulin sensitizing in cells. Diabetic mice treated with azilsartan had lowered expressions of pro-inflammatory cytokines in brain vessels and lowered diabetes-induced BBB permeability.

Product Info

Cas No.

863031-21-4

Purity

≥98%

Formula

C30H24N4O8

Formula Wt.

568.54

Chemical Name

1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic Acid (5-Methyl-2-oxo-1,3-dioxol-4-yl)methyl ester

IUPAC Name

(5-methyl-2-oxo-1,3-dioxol-4-yl)methyl 2-ethoxy-3-[[4-[2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]phenyl]methyl]benzimidazole-4-carboxylate

Synonym

TAK 491; TAK-491; TAK491

Melting Point

212-214

Shipping and Storage

Store Temp

-20°C

Ship Temp

Ambient

Downloads

MSDS

A971336 MSDS PDF

Info Sheet

A971336 Info Sheet PDF

References

Kurtz T, Kajiya T. Differential pharmacology and benefit/risk of azilsartan compared to other sartans. Vasc Health Risk Manag. 2012;8:133-143. PMID: 22399858.

Han J, Tang H, Yao L, et al. Azilsartan protects against hyperglycemia-induced hyperpermeability of the blood-brain barrier. Bioengineered. 2021 Dec;12(1):3621-3633. PMID: 34266350.

Li W, Wang C, Zhang D, et al. Azilsartan ameliorates ox-LDL-induced endothelial dysfunction via promoting the expression of KLF2. Aging (Albany NY). 2021 May 4; 13(9):12996-13005. PMID: 33946046.

Baker W, White W. Azilsartan medoxomil: a new angiotensin II receptor antagonist for treatment of hypertension. Ann Pharmacother. 2011 Dec;45(12):1506-1515. PMID: 22116996.

Custom Order

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