LKT Labs

Biochemicals for Life Science Research

KB-0742

KB-0742

Product ID K040007
Cas No. 2170137-61-6 (free base)
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $204.00 In stock
5 mg $403.00 In stock
10 mg $606.00 In stock
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Description

KB-0742 is a selective CDK9 inhibitor with potent anti-tumor activity in castration-resistant prostate cancer models.

Product Info

Cas No.

2170137-61-6 (free base)
Purity

≥98%
Formula

C16H25N5
Formula Wt.

287.41
IUPAC Name

(1S,3S)-3-N-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamine
Synonym

KB0742, NSC-834161, NSC834161
Appearance

Yellow to brown crystal

Shipping and Storage

Store Temp

-20°C
Ship Temp

Ambient

Downloads

Info Sheet

K040007 Info Sheet PDF

References

Richters A, Doyle S, Freeman D, et al. Modulating androgen receptor-driven transcription in prostate cancer with selective CDK9 inhibitors. Cell Chem Biol. 2021 Feb 18;28(2):134-147. PMID: 33086052

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