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Flumazenil

Flumazenil

Product ID F4681
Cas No. 78755-81-4
Purity ≥98%
Product Unit SizeCostQuantityStock
5 mg $75.10 In stock
25 mg $147.20 In stock
100 mg $443.30 In stock
Bulk Quote

Quicklinks

  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Description
  • Product Info
  • Shipping and Storage
  • Downloads
  • References
  • Custom Order

Description

Flumazenil is an antagonist at GABA-A receptors that is used as a stimulant to counteract the effects of benzodiazepines. Flumenazil inhibits benzodiazepine-induced sedation, motor impairment, and ventilator depression.

Product Info

Cas No.

78755-81-4

Purity

≥98%

Formula

C15H14FN3O3

Formula Wt.

303.29

Chemical Name

8-Fluoro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepinne-3-carboxylic acid ethyl ester

IUPAC Name

ethyl 8-fluoro-5-methyl-6-oxo-4H-imidazo[1,5-a][1, 4]benzodiazepine-3-carboxylate

Synonym

Anexate, Ro-15-1788, Lanexat, Romazicon

Melting Point

201-203°C

Solubility

Soluble in water (128mg/L).

Appearance

A white or almost white crystalline powder

Shipping and Storage

Store Temp

4°C

Ship Temp

Ambient

Downloads

MSDS

F4681 MSDS PDF

Info Sheet

F4681 Info Sheet PDF

References

Rye DB, Bliwise DL, Parker K, et al. Modulation of vigilance in the primary hypersomnias by endogenous enhancement of GABAA receptors. Sci Transl Med. 2012 Nov 21;4(161):161ra151. PMID: 23175709.

Lader M. Benzodiazepines revisited--will we ever learn? Addiction. 2011 Dec;106(12):2086-109. PMID: 21714826.

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
  • Total quantity of unit size desired (e.g. '10' in the case of 10 x 500 mg). If only one unit is desired, you may leave this blank.
  • This field is for validation purposes and should be left unchanged.

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